SCHEMBL7323557

SCHEMBL7323557

CCOC(=O)c1ccc(OC(Cc2ccccc2)Cc2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.57
PPARG P37231 6/20 0.52
PPARA Q07869 5/20 0.52
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
MAPT P10636 2/20 0.50
NAMPT P43490 1/20 0.50
LMNA P02545 2/20 0.49
GAA P10253 2/20 0.49
RAB9A P51151 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
NPC1 O15118 1/20 0.49
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
ESR1 P03372 1/20 0.49
CA7 P43166 1/20 0.49
CA9 Q16790 1/20 0.49
ESR2 Q92731 1/20 0.49
CA14 Q9ULX7 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7324691 0.82 NR4A1 (0.57) PPARGPPARAKMT2A
SCHEMBL119521 0.79 SRD5A2 (0.59) SMN1; SMN2PPARGMEN1KMT2AMAPT
SCHEMBL7314137 0.79 PPARG (0.52) PPARGPPARA
SCHEMBL9818904 0.79 RAB9A (0.52) SMN1; SMN2PPARGPPARAKMT2AMAPT
SCHEMBL10487454 0.78 RAB9A (0.51) SMN1; SMN2PPARGPPARAMEN1KMT2A
SCHEMBL340618 0.78 MAOB (0.67) SMN1; SMN2PPARGKMT2AMAPTLMNA
SCHEMBL7322562 0.78 SMN1; SMN2 (0.51) SMN1; SMN2MEN1KMT2AMAPTNAMPT
Benzene SCHEMBL27873122 0.78 CA1 (0.76) SMN1; SMN2MEN1KMT2AMAPTLMNA
SCHEMBL9597273 0.77 FFAR1 (0.48) SMN1; SMN2LMNARAB9AL3MBTL1NPC1
SCHEMBL9597276 0.77 FFAR1 (0.48) SMN1; SMN2LMNARAB9AL3MBTL1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0927035-A4 THROMBIN INHIBITORS MERCK & CO INC (US) 2002-11-13 EP disclosed
EP-0927035-A1 THROMBIN INHIBITORS Merck & Co., Inc. (US) 1999-07-07 EP disclosed
US-5872138-A INHIBITING LOSS OF BLOOD PLATELETS, INHIBITING FORMATION OF BLOOD PLATELET AGGREGATES, INHIBITING FORMATION OF FIBRIN, INHIBITING THROMBUS FORMATION, AND INHIBITING EMBOLUS FORMATION IN A MAMMAL MERCK & CO., INC. (US) 1999-02-16 US disclosed
WO-1998010763-A1 THROMBIN INHIBITORS MERCK & CO., INC. (US) 1998-03-19 WO disclosed