SCHEMBL7323606

SCHEMBL7323606

CCOC(OCC)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)C(C)C

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CMA1 P23946 5/20 0.53
ELANE P08246 7/20 0.51
CAPN1 P07384 2/20 0.51
CTSL P07711 1/20 0.50
CTSB P07858 1/20 0.50
CTSK P43235 1/20 0.50
MALT1 Q9UDY8 1/20 0.49
PREP P48147 2/20 0.49
CCR1 P32246 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7285949 1.00 CMA1 (0.53) CMA1ELANECAPN1CTSLCTSB
SCHEMBL7320477 0.92 CMA1 (0.53) CMA1ELANEMALT1
SCHEMBL7316337 0.90 MALT1 (0.59) CMA1ELANECTSLMALT1PREP
SCHEMBL7355181 0.88 MALT1 (0.59) CMA1ELANEMALT1
SCHEMBL7311225 0.86 DPP8 (0.52) CMA1ELANEMALT1
Hydrochloric Acid SCHEMBL7287630 0.86 CMA1 (0.50) CMA1ELANECAPN1CTSLCTSB
SCHEMBL13036085 0.86 CMA1 (0.55) CMA1ELANEMALT1
SCHEMBL10080680 0.86 ELANE (0.57) CMA1ELANECAPN1CTSLCTSB
SCHEMBL7279072 0.85 CTSL (0.56) CMA1ELANECAPN1CTSLCTSB
SCHEMBL8092357 0.85 CMA1 (0.58) CMA1ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4923890-A Difluoro keto compounds and their use as HLE inhibitors ICI AMERICAS INC. (US) 1990-05-08 US disclosed
EP-0249349-A1 Difluoroketo compounds ICI AMERICAS INC. (US) 1987-12-16 EP disclosed
US-4691007-A HUMAN LEUKOCYTE ELASTASE INHIBITORS ICI AMERICAS INC. (US) 1987-09-01 US disclosed
EP-0204571-A2 Selected difluoro derivatives ICI AMERICAS INC. (US) 1986-12-10 EP disclosed
US-4596789-A Pharmaceuticals ICI AMERICAS INC. (US) 1986-06-24 US disclosed
EP-0124317-A2 Proline derivatives ICI AMERICAS INC. (US) 1984-11-07 EP disclosed