SCHEMBL7325147

SCHEMBL7325147

COC(=O)c1cc(Cl)c(NC(C)=O)c2c1OCCCC2

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.36
KDM4E B2RXH2 4/20 0.36
MAPK1 P28482 1/20 0.36
SMN1; SMN2 Q16637 4/20 0.36
HPGD P15428 2/20 0.36
MAPT P10636 1/20 0.36
HSD17B10 Q99714 1/20 0.34
GAA P10253 1/20 0.34
ACHE P22303 1/20 0.34
NQO2 P16083 1/20 0.33
TSHR P16473 1/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
KMT2A Q03164 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8690082 0.96 KDM4E (0.37) ALDH1A1KDM4EMAPK1SMN1; SMN2HPGD
SCHEMBL6600592 0.91 HTR4 (0.38) ALDH1A1KDM4EMAPK1SMN1; SMN2GAA
SCHEMBL7386673 0.84 HSD17B10 (0.40) ALDH1A1KDM4EMAPK1HPGDHSD17B10
SCHEMBL5315483 0.82 KDM4E (0.35) ALDH1A1KDM4EMAPK1SMN1; SMN2HPGD
SCHEMBL7324275 0.81 ALDH1A1 (0.35) ALDH1A1KDM4EMAPK1SMN1; SMN2HPGD
SCHEMBL7325188 0.81 KDM4E (0.34) ALDH1A1KDM4EMAPK1SMN1; SMN2HPGD
SCHEMBL8500298 0.80 HTR4 (0.36) ALDH1A1KDM4EHSD17B10ACHE
SCHEMBL6586553 0.79 KDM4E (0.41) ALDH1A1KDM4EMAPK1HSD17B10ACHE
SCHEMBL8132698 0.78 MAPK1 (0.36) ALDH1A1KDM4EMAPK1SMN1; SMN2HPGD
SCHEMBL14810317 0.78 HTR4 (0.48) ALDH1A1KDM4EGAAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4924010-A GASTROINTESTINAL DISORDERS RORER PHARMACEUTICAL CORPORATION (US) 1990-05-08 US disclosed
US-4859683-A Certain benzoxepins and their pharmaceutical compositions and methods RORER PHARMACEUTICAL CORPORATION (US) 1989-08-22 US disclosed
US-4857517-A Quinuclidyl benzoxepins as 5-HT3 antagonists RORER PHARMACEUTICAL CORPORATION (US) 1989-08-15 US disclosed