SCHEMBL7325537

SCHEMBL7325537

CCCc1[nH]cnc1C(C)=C(C)C(N)=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.39
HSD17B10 Q99714 1/20 0.39
LMNA P02545 1/20 0.36
GABRR1 P24046 1/20 0.36
KDM4E B2RXH2 1/20 0.35
HRH2 P25021 1/20 0.34
HRH1 P35367 1/20 0.34
HRH4 Q9H3N8 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
XDH P47989 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
GDA Q9Y2T3 1/20 0.32
PDE4A P27815 2/20 0.32
PDE4B Q07343 2/20 0.32
PDE4C Q08493 2/20 0.32
PDE4D Q08499 2/20 0.32
GAA P10253 3/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
USP2 O75604 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6499135 0.82 CYP2C19 (0.44) CYP2C19HSD17B10LMNAKDM4EXDH
SCHEMBL5870589 0.76 CYP2C19 (0.65) CYP2C19HSD17B10LMNAGABRR1KDM4E
SCHEMBL5870372 0.75 CYP2C19 (0.44) CYP2C19HSD17B10LMNAGABRR1KDM4E
Hydrochloric Acid SCHEMBL5869997 0.75 CYP2C19 (0.62) CYP2C19HSD17B10LMNAGABRR1KDM4E
SCHEMBL2101530 0.72 LMNA (0.45) CYP2C19HSD17B10LMNAKDM4EHRH3
SCHEMBL5870375 0.72 SMN1; SMN2 (0.42) CYP2C19HSD17B10LMNAKDM4ETDP1
SCHEMBL5870445 0.71 KDM4E (0.58) HSD17B10LMNAKDM4EGAASMN1; SMN2
SCHEMBL5870451 0.71 HPGD (0.41) CYP2C19HSD17B10KDM4EGAASMN1; SMN2
SCHEMBL6500732 0.69 CYP2C19 (0.46) CYP2C19HSD17B10LMNAGABRR1KDM4E
SCHEMBL14692540 0.68 CYP2C19 (0.57) CYP2C19HSD17B10LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0242973-B1 INDOLE DERIVATIVES, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1991-07-17 EP disclosed