SCHEMBL7325663

SCHEMBL7325663

CN(CCc1ccoc1)C1CCc2c(N)cccc2C1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 11/20 0.42
DRD1 P21728 7/20 0.42
DRD3 P35462 5/20 0.40
DRD4 P21917 4/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
NFKB1 P19838 1/20 0.40
THPO P40225 1/20 0.40
LMNA P02545 1/20 0.39
PMP22 Q01453 1/20 0.39
HTR1A P08908 3/20 0.39
HTR7 P34969 3/20 0.39
DRD5 P21918 1/20 0.38
ADRB2 P07550 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7329471 0.94 GRIN2B (0.40) DRD2DRD1DRD3HTR1AHTR7
SCHEMBL7328341 0.93 GRIN2B (0.41) DRD2DRD1DRD3
SCHEMBL7328585 0.92 DRD2 (0.41) DRD2DRD1DRD3
SCHEMBL7332957 0.89 HTR1A (0.40) DRD2DRD1DRD3DRD4HTR1A
SCHEMBL7327614 0.87 DRD2 (0.50) DRD2DRD1DRD3DRD4CYP1A2
SCHEMBL7325610 0.85 DRD2 (0.54) DRD2DRD1DRD3DRD4CYP1A2
SCHEMBL7329557 0.83 DRD2 (0.47) DRD2DRD1DRD3DRD4HTR1A
SCHEMBL7330395 0.82 DRD2 (0.47) DRD2DRD1DRD3DRD4HTR1A
SCHEMBL7333718 0.82 DRD2 (0.46) DRD2DRD1DRD3DRD4CYP1A2
SCHEMBL7328110 0.81 DRD2 (0.48) DRD2DRD1DRD3DRD4HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0402923-A2 2,5-Diaminotetralines, process for their preparation and their use as medicine BOEHRINGER INGELHEIM KG (DE) 1990-12-19 EP disclosed