SCHEMBL7325664

SCHEMBL7325664

NC(=O)c1cccc(CO)c1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGB1 P09429 1/20 0.49
KDM4E B2RXH2 3/20 0.47
HPGD P15428 2/20 0.47
ALDH1A1 P00352 2/20 0.47
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.47
HSD17B10 Q99714 1/20 0.47
PARP1 P09874 4/20 0.46
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
BCAT2 O15382 1/20 0.42
GABRA1 P14867 1/20 0.40
GABRB2 P47870 1/20 0.40
GAA P10253 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
CXCR2 P25025 1/20 0.40
LMNA P02545 1/20 0.40
METAP2 P50579 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
MMP2 P08253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7727117 0.84 GABRA1 (0.61) HMGB1KDM4EHPGDALDH1A1MAPT
SCHEMBL16585595 0.84 HMGB1 (0.53) HMGB1KDM4EHPGDALDH1A1MAPT
SCHEMBL28593606 0.82 HMGB1 (0.65) HMGB1KDM4EHPGDALDH1A1HSD17B10
SCHEMBL27733222 0.82 ERN1 (0.42) KDM4EHPGDALDH1A1MAPTTSHR
SCHEMBL619877 0.81 ALDH1A1 (0.52) KDM4EHPGDALDH1A1MAPTTSHR
SCHEMBL698742 0.80 KDM4E (0.61) KDM4EHPGDALDH1A1MAPTTSHR
SCHEMBL5545298 0.80 PARP1 (0.46) KDM4EHPGDALDH1A1MAPTTSHR
SCHEMBL2129165 0.80 PARP1 (0.46) HMGB1KDM4EHPGDALDH1A1MAPT
Ammonia Solution, Strong SCHEMBL27393517 0.79 ALDH1A1 (0.50) KDM4EHPGDALDH1A1MAPTTSHR
SCHEMBL2896616 0.78 PARP1 (0.44) KDM4EHPGDALDH1A1MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0271059-B1 2-Methylthiomethyl-dihydropyridines, a process for their preparation and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA (IT) 1993-10-20 EP disclosed
US-4971984-A Cardiovascular disorders, hypotensive agints BEEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1990-11-20 US disclosed