SCHEMBL7325705

SCHEMBL7325705

CN1CCN(c2cc(=O)c3ccccc3o2)CC1

nearest known ligand 0.71

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 14/20 0.71
ACE P12821 1/20 0.71
ECE1 P42892 1/20 0.71
TNKS O95271 1/20 0.52
XRCC6 P12956 1/20 0.51
XRCC5 P13010 1/20 0.51
P2RY12 Q9H244 1/20 0.50
MAOB P27338 1/20 0.47
HRH4 Q9H3N8 2/20 0.46
PIK3R1 P27986 1/20 0.46
PIK3CA P42336 1/20 0.46
MTOR P42345 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A1 P04798 1/20 0.45
CYP1B1 Q16678 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31035740 0.84 PRKDC (0.75) PRKDCACEECE1XRCC6XRCC5
SCHEMBL30218216 0.83 PRKDC (1.00) PRKDCACEECE1XRCC6XRCC5
SCHEMBL3361567 0.83 PRKDC (1.00) PRKDCACEECE1XRCC6XRCC5
SCHEMBL25246006 0.82 PRKDC (0.71) PRKDCACEECE1XRCC6XRCC5
SCHEMBL5476610 0.82 PRKDC (0.71) PRKDCACEECE1XRCC6XRCC5
SCHEMBL3538463 0.79 PRKDC (0.78) PRKDCPIK3R1PIK3CAMTORTDP1
SCHEMBL7294524 0.75 SIGMAR1 (0.76) PRKDCACEECE1TNKSALDH1A1
SCHEMBL14081448 0.74 TNKS (0.47) PRKDCACEECE1TNKSMAOB
SCHEMBL8788233 0.72 ACE (0.58) PRKDCACEECE1TNKSMAOB
SCHEMBL7324233 0.72 HTR6 (0.56) PRKDCXRCC6XRCC5HRH4PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5703075-A Antiatherosclerotic and antithrombotic 1-benzopyran-4-ones and 2-amino-1,3-benzoxazine-4-ones PHARMACIA & UPJOHN COMPANY (US) 1997-12-30 US disclosed
EP-0459983-A1 ANTIATHEROSCLEROTIC AND ANTITHROMBOTIC 1-BENZOPYRAN-4-ONES AND 2-AMINO-1,3-BENZOXAZINE-4-ONES PHARMACIA & UPJOHN COMPANY (US) 1991-12-11 EP disclosed
WO-1990006921-A1 ANTIATHEROSCLEROTIC AND ANTITHROMBOTIC 1-BENZOPYRAN-4-ONES AND 2-AMINO-1,3-BENZOXAZINE-4-ONES THE UPJOHN COMPANY (US) 1990-06-28 WO disclosed