SCHEMBL7326223

SCHEMBL7326223

COc1ccc(CCCNCCC(=O)Nc2ccc(F)cc2)cc1OC

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
ALDH1A1 P00352 1/20 0.52
CNR1 P21554 1/20 0.52
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
HDAC1 Q13547 2/20 0.52
HDAC2 Q92769 2/20 0.52
ATM Q13315 1/20 0.52
EPHX2 P34913 1/20 0.51
GAA P10253 1/20 0.49
THRB P10828 1/20 0.49
ADRB2 P07550 1/20 0.48
ADRB1 P08588 1/20 0.48
ADRB3 P13945 1/20 0.48
MAPT P10636 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7359187 0.85 KMT2A (0.58) NPC1RAB9AALDH1A1CNR1MEN1
SCHEMBL7360125 0.85 NPC1 (0.55) NPC1RAB9AALDH1A1CNR1MEN1
SCHEMBL7335367 0.83 NPC1 (0.55) NPC1RAB9AALDH1A1CNR1HDAC1
SCHEMBL7356345 0.81 NPC1 (0.65) NPC1RAB9AHDAC1HDAC2
SCHEMBL7326215 0.80 CYP3A4 (0.67) NPC1RAB9AALDH1A1MEN1KMT2A
SCHEMBL7175921 0.80 PLAAT3 (0.54) MEN1KMT2AHDAC1HDAC2ATM
SCHEMBL7331861 0.80 PLAAT3 (0.57) ALDH1A1HDAC1HDAC2ATMSMN1; SMN2
SCHEMBL7355959 0.78 HDAC1 (0.54) NPC1RAB9AALDH1A1MEN1KMT2A
SCHEMBL18760165 0.77 NPC1 (0.67) NPC1RAB9AALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL9782076 0.76 SLC2A1 (0.65) ALDH1A1KMT2AATMADRB2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0852142-A1 Diamines in the treatment of arrhythmia SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1998-07-08 EP disclosed
EP-0639973-A1 DIAMINES IN THE TREATMENT OF ARRHYTHMIA SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1995-03-01 EP disclosed
WO-1993023024-A1 DIAMINES IN THE TREATMENT OF ARRHYTHMIA SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1993-11-25 WO disclosed