SCHEMBL7335367

SCHEMBL7335367

COc1ccc(CCCNCCC(=O)Nc2ccc(OC(C)C)c(OC(C)C)c2)cc1OC

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
HDAC1 Q13547 5/20 0.50
HDAC2 Q92769 5/20 0.50
LMNA P02545 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CNR1 P21554 1/20 0.46
GAA P10253 1/20 0.45
PKM P14618 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
EPHX2 P34913 1/20 0.45
POLB P06746 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC8 Q9BY41 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7359187 0.84 KMT2A (0.58) NPC1RAB9AHDAC1HDAC2LMNA
SCHEMBL7360125 0.83 NPC1 (0.55) NPC1RAB9AHDAC1HDAC2LMNA
SCHEMBL7326223 0.83 NPC1 (0.54) NPC1RAB9AHDAC1HDAC2SMN1; SMN2
SCHEMBL7356345 0.82 NPC1 (0.65) NPC1RAB9AHDAC1HDAC2POLB
SCHEMBL7335360 0.82 CYP3A4 (0.62) NPC1RAB9AHDAC1HDAC2LMNA
SCHEMBL7355959 0.79 HDAC1 (0.54) NPC1RAB9AHDAC1HDAC2LMNA
SCHEMBL18760165 0.78 NPC1 (0.67) NPC1RAB9AHDAC1HDAC2LMNA
SCHEMBL7331861 0.76 PLAAT3 (0.57) HDAC1HDAC2SMN1; SMN2POLBKDM4E
SCHEMBL7175921 0.76 PLAAT3 (0.54) HDAC1HDAC2SMN1; SMN2POLBKDM4E
SCHEMBL7355352 0.73 LMNA (0.56) NPC1RAB9AHDAC1HDAC2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0852142-A1 Diamines in the treatment of arrhythmia SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1998-07-08 EP disclosed
EP-0639973-A1 DIAMINES IN THE TREATMENT OF ARRHYTHMIA SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1995-03-01 EP disclosed
WO-1993023024-A1 DIAMINES IN THE TREATMENT OF ARRHYTHMIA SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1993-11-25 WO disclosed