SCHEMBL7326419

SCHEMBL7326419

CCc1ccccc1/C=C/CBr

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.40
GABRB2 P47870 2/20 0.40
PTGER3 P43115 5/20 0.37
PTGER2 P43116 5/20 0.37
PTGER4 P35408 4/20 0.37
PTGER1 P34995 2/20 0.37
CHAT P28329 1/20 0.37
TSHR P16473 2/20 0.34
CYP2D6 P10635 2/20 0.33
MGLL Q99685 1/20 0.33
TBXA2R P21731 1/20 0.33
PTGDR Q13258 1/20 0.33
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC11 Q96DB2 1/20 0.32
HDAC8 Q9BY41 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28412294 0.83 PTGER3 (0.39) GABRA1GABRB2PTGER3PTGER2PTGER4
SCHEMBL6546259 0.83 CHAT (0.47) GABRA1GABRB2PTGER3PTGER2PTGER4
SCHEMBL3314625 0.83 CHAT (0.47) GABRA1GABRB2PTGER3PTGER2PTGER4
SCHEMBL17155197 0.80 PTGER3 (0.37) GABRA1GABRB2PTGER3PTGER2PTGER4
SCHEMBL5892736 0.79 GABRA1 (0.43) GABRA1GABRB2TSHRCYP2D6MGLL
SCHEMBL5033527 0.77 PDE5A (0.43) PTGER3PTGER2PTGER4PTGER1TSHR
SCHEMBL6546515 0.77 MAOB (0.50) PTGER3PTGER2PTGER4PTGER1CHAT
SCHEMBL6546519 0.77 MAOB (0.50) PTGER3PTGER2PTGER4PTGER1CHAT
SCHEMBL9494233 0.77 CHAT (0.40) GABRA1GABRB2PTGER3PTGER2PTGER4
SCHEMBL31094912 0.77 CHAT (0.40) GABRA1GABRB2PTGER3PTGER2PTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0347766-A2 4,5,7,8-Tetrahydro-6H-thiazolo[5,4-d]azepines, their preparation and their use as medicaments Dr. Karl Thomae GmbH (DE) 1989-12-27 EP disclosed