SCHEMBL7326626

SCHEMBL7326626

O=CCCN1C(=O)c2cccc3cccc(c23)C1=O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HEXA P06865 6/20 0.68
HEXB P07686 6/20 0.68
OGA O60502 1/20 0.68
SIRT1 Q96EB6 3/20 0.62
KDM4E B2RXH2 3/20 0.59
ALDH1A1 P00352 3/20 0.59
MAPT P10636 2/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
GAA P10253 1/20 0.59
RAB9A P51151 1/20 0.59
CYP1B1 Q16678 1/20 0.59
KMT2A Q03164 3/20 0.56
MEN1 O00255 2/20 0.56
POLB P06746 2/20 0.56
NR1I2 O75469 1/20 0.56
AHR P35869 1/20 0.56
RAD52 P43351 1/20 0.56
RCE1 Q9Y256 1/20 0.56
HSD17B10 Q99714 2/20 0.54
HPGD P15428 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7324978 0.90 HEXA (0.67) HEXAHEXBOGASIRT1KDM4E
SCHEMBL1042197 0.83 GLS (0.57) MAPTSMN1; SMN2RAB9ACYP1A2
SCHEMBL30185439 0.83 GLS (0.57) MAPTSMN1; SMN2RAB9ACYP1A2
SCHEMBL7319904 0.82 CYP1B1 (0.62) HEXAHEXBOGASIRT1KDM4E
SCHEMBL9626265 0.82 HEXA (0.83) HEXAHEXBOGASIRT1KDM4E
SCHEMBL4408773 0.81 HEXA (1.00) HEXAHEXBOGASIRT1KDM4E
SCHEMBL31011151 0.81 HEXA (1.00) HEXAHEXBOGASIRT1KDM4E
SCHEMBL9625535 0.80 HEXA (0.81) HEXAHEXBOGASIRT1KDM4E
SCHEMBL9625779 0.80 HEXA (0.81) HEXAHEXBOGASIRT1KDM4E
SCHEMBL9625518 0.80 HEXA (0.81) HEXAHEXBOGASIRT1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995013817-A1 ENDOTHELIN CONVERTING ENZYME INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1995-05-26 WO disclosed
EP-0612324-A1 PHOSPHONOPEPTIDES WITH COLLAGENASE INHIBITING ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1994-08-31 EP disclosed
WO-1993009136-A1 PHOSPHONOPEPTIDES WITH COLLAGENASE INHIBITING ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1993-05-13 WO disclosed