SCHEMBL7327907

SCHEMBL7327907

COC(=O)[C@H](Cc1c[nH]cn1)N(C)C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 1/20 0.36
AAK1 Q2M2I8 4/20 0.35
TDP1 Q9NUW8 6/20 0.33
POLB P06746 4/20 0.33
NPSR1 Q6W5P4 3/20 0.33
MAPT P10636 3/20 0.33
ATM Q13315 2/20 0.32
HCRTR1 O43613 1/20 0.32
XBP1 P17861 1/20 0.31
RECQL P46063 1/20 0.31
REN P00797 1/20 0.31
TACR1 P25103 1/20 0.31
ADORA1 P30542 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8189733 0.89 TDP1 (0.34) TDP1POLBNPSR1MAPTATM
SCHEMBL7325648 0.86 AAK1 (0.37) MMP13AAK1TDP1POLBNPSR1
SCHEMBL9847303 0.84 SIRT2 (0.31)
SCHEMBL12199030 0.82 MAPK1 (0.33) TACR1ALDH1A1
SCHEMBL14324686 0.82 MAPK1 (0.33) TACR1ALDH1A1
Hydrochloric Acid SCHEMBL8183614 0.81 ALDH1A1 (0.33) MAPTTACR1ALDH1A1
SCHEMBL3341580 0.81 ADORA1 (0.37) MMP13TDP1NPSR1MAPTATM
SCHEMBL7328213 0.80 ABCB1 (0.47) MAPTRECQLALDH1A1
SCHEMBL6833631 0.79 TDP1 (0.33) TDP1POLBNPSR1MAPTATM
SCHEMBL4891567 0.79 TDP1 (0.33) TDP1POLBNPSR1MAPTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0396065-A1 Novel amino acid derivatives possessing renin-inhibitory activities Japan Tobacco Inc. (JP) 1990-11-07 EP disclosed