SCHEMBL7328213

SCHEMBL7328213

COC(=O)[C@H](Cc1c[nH]cn1)N(C)C(=O)OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.47
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
CTSK P43235 2/20 0.39
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
CTSS P25774 1/20 0.39
ALDH1A1 P00352 2/20 0.39
TRPM8 Q7Z2W7 1/20 0.39
ALOX15 P16050 1/20 0.39
CTRB1 P17538 2/20 0.39
MAPT P10636 1/20 0.38
RECQL P46063 1/20 0.38
EPOR P19235 1/20 0.37
LTA4H P09960 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7333726 0.89 ABCB1 (0.43) ABCB1ITGB3ITGA2BCTSKCTSL
SCHEMBL10436050 0.83 CIT (0.41) ABCB1ALDH1A1ALOX15LTA4H
SCHEMBL9847303 0.82 SIRT2 (0.31)
SCHEMBL22457646 0.82 ABCB1 (0.62) ABCB1ITGB3ITGA2BCTSKCTSL
SCHEMBL11639032 0.82 CTRB1 (0.39) ABCB1ITGB3ITGA2BALDH1A1CTRB1
SCHEMBL11267790 0.81 ABCB1 (0.37) ABCB1ALDH1A1TRPM8ALOX15CTRB1
SCHEMBL29897717 0.80 CTRB1 (0.38) ABCB1ITGB3ITGA2BALDH1A1CTRB1
SCHEMBL7327907 0.80 MMP13 (0.36) ALDH1A1MAPTRECQL
SCHEMBL6371254 0.79 EPOR (0.35) ALDH1A1TRPM8ALOX15CTRB1MAPT
SCHEMBL29401219 0.79 ALDH1A1 (0.54) CTSKCTSLCTSBCTSSALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0396065-A1 Novel amino acid derivatives possessing renin-inhibitory activities Japan Tobacco Inc. (JP) 1990-11-07 EP disclosed