SCHEMBL7328733

SCHEMBL7328733

COC(OC)c1ccc(CBr)cc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.39
TRPA1 O75762 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
IDO1 P14902 2/20 0.33
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
CA2 P00918 1/20 0.31
L3MBTL1 Q9Y468 2/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
MAPK1 P28482 1/20 0.30
ATM Q13315 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL450723 0.89 TRPA1 (0.31) TSHRTRPA1ALDH1A1
SCHEMBL15953591 0.83 TDP1 (0.43) CYP1A2CYP2D6CYP2C19IDO1TDP1
SCHEMBL8955219 0.80 CA12 (0.35) TSHRALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL9008790 0.79 TDP1 (0.50) TSHRALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL6947245 0.78 ACHE (0.46) TSHRTRPA1ALDH1A1IDO1CES2
SCHEMBL8954887 0.77 IDO1 (0.42) CYP1A2CYP2D6CYP2C19IDO1CA2
SCHEMBL7349245 0.77 HRH3 (0.44) CYP1A2CYP2D6CYP2C19IDO1
SCHEMBL19640126 0.77 TTR (0.37) TSHRCYP1A2CYP2D6CYP2C19IDO1
SCHEMBL2938648 0.77 LTA4H (0.39) TSHRCYP1A2CYP2D6CYP2C19IDO1
SCHEMBL11249724 0.76 PTGS1 (0.50) TSHRESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014203132-A1 SUBSTITUTED BENZOPYRAN COMPOUNDS, COMPOSITIONS AND USES THEREOF OLEMA PHARMACEUTICALS, INC. (US) 2014-12-24 WO disclosed
US-20090023842-A1 PORPHYRIN AND CONDUCTIVE POLYMER COMPOSITIONS FOR USE IN SOLID-STATE ELECTRONIC DEVICES PLEXTRONICS, INC. 2009-01-22 US disclosed
US-20090023842-A1 PORPHYRIN AND CONDUCTIVE POLYMER COMPOSITIONS FOR USE IN SOLID-STATE ELECTRONIC DEVICES PLEXTRONICS, INC. 2009-01-22 US disclosed
WO-2008144750-A1 PORPHYRIN AND CONDUCTIVE POLYMER COMPOSITIONS FOR USE IN SOLID-STATE ELECTRONIC DEVICES PLEXTRONICS, INC. (US) 2008-11-27 WO disclosed
EP-0434365-A2 HIV protease inhibitors useful for the treatment of aids MERCK & CO. INC. (US) 1991-06-26 EP disclosed
EP-0145263-B1 LIVING POLYMERS AND PROCESS FOR THEIR PREPARATION E.I. DU PONT DE NEMOURS AND COMPANY (US) 1991-04-17 EP disclosed
US-4783500-A ORGANO-SILICON,-TIN, OR -GERMANIUM INITIATORS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1988-11-08 US disclosed
US-4711942-A FROM ACRYLIC OR MALEIMIDE MONOMER AND ORGANOSILICON,-TIN, OR -GERMANIUM INITIATOR E. I. DU PONT DE NEMOURS AND COMPANY (US) 1987-12-08 US disclosed
US-4681918-A ACRYLIC-TYPE OR MALEIMIDE MONOMERS; ORGANOSILICON, TIN OR GERMANIUM INITIATORS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1987-07-21 US disclosed
EP-0068887-B1 \"LIVING\" POLYMERS AND PROCESS FOR THEIR PREPARATION E.I. DU PONT DE NEMOURS AND COMPANY (US) 1986-09-24 EP disclosed
US-4581428-A Process for preparing \"living\" polymers using tetracoordinate organosilicon, organotin or organogermanium polymerization initiator with bifluoride ion source co-catalyst E. I. DU PONT DE NEMOURS AND COMPANY (US) 1986-04-08 US disclosed
EP-0145263-A1 Living polymers and process for their preparation E.I. DU PONT DE NEMOURS AND COMPANY (US) 1985-06-19 EP disclosed
US-4524196-A Process for preparing \"living\" polymers E. I. DU PONT DE NEMOURS AND COMPANY (US) 1985-06-18 US disclosed
US-4508880-A ACRYLIC OR MALEIMIDE MONOMERS WITH ORGANOSILICON, (-TIN, OR-GERMANIUM) INITIATORS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1985-04-02 US disclosed
US-4417034-A POLYMERIZING ACRYLIC OR MALEIMIDE MONOMERS WITH ORGANO-SILICON, -TIN, OR-GERMANIUM INITIATORS E. I. DU PONT DE NEMOURS & CO. (US) 1983-11-22 US disclosed
US-4414372-A ADDITION POLYMERS WITH FUNCTIONAL END GROUPS E. I. DU PONT DE NEMOURS & CO. (US) 1983-11-08 US disclosed
EP-0068887-A1 \"Living\" polymers and process for their preparation E.I. DU PONT DE NEMOURS AND COMPANY (US) 1983-01-05 EP disclosed