SCHEMBL7329079

SCHEMBL7329079

CCCCS(=O)(=O)N[C@@H](CC1=CCC(O)(CCCC(=O)c2nc3ccccc3[nH]2)C=C1)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DAGLA Q9Y4D2 2/20 0.44
ITGB3 P05106 12/20 0.37
ITGA2B P08514 10/20 0.37
PIN1 Q13526 2/20 0.35
ITGAV P06756 3/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SPHK2 Q9NRA0 1/20 0.35
SPHK1 Q9NYA1 1/20 0.35
CHRM2 P08172 1/20 0.34
SLC6A4 P31645 1/20 0.34
SMYD3 Q9H7B4 1/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7329238 0.81 ALDH1A1 (0.40) PIN1NPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL27573148 0.68 DAGLA (0.76) DAGLANPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL7542370 0.66 BCHE (0.43) ITGB3ITGA2BPIN1ITGAVNPC1
SCHEMBL7347037 0.65 ALDH1A1 (0.56) DAGLAPIN1NPC1ALDH1A1RAB9A
SCHEMBL7347042 0.65 ALDH1A1 (0.56) DAGLAPIN1NPC1ALDH1A1RAB9A
SCHEMBL6032775 0.64 ITGB3 (0.64) ITGB3ITGA2BITGAVALDH1A1CHRM2
SCHEMBL7329235 0.64 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2
SCHEMBL3962735 0.63 DAGLA (1.00) DAGLANPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL5603960 0.62 ITGB3 (0.61) ITGB3ITGA2BITGAVALDH1A1CHRM2
SCHEMBL7622370 0.62 ITGB3 (0.61) ITGB3ITGA2BITGAVALDH1A1CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0767792-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2002-11-20 EP disclosed
US-5977101-A Benzimidazoles/Imidazoles Linked to a Fibrinogen Receptor Antagonist Template Having Vitronectin Receptor Antagonist Activity SMITHKLINE BEECHAM CORPORATION (US) 1999-11-02 US disclosed
EP-0767792-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-04-16 EP disclosed
WO-1996000730-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1996-01-11 WO disclosed