SCHEMBL7542370

SCHEMBL7542370

CCCCS(=O)(=O)NC(Cc1ccc2c(c1)Cc1cc(CCNc3nc4ccccc4[nH]3)ccc1-2)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.43
TRPC3 Q13507 1/20 0.43
TRPC4 Q9UBN4 1/20 0.43
TRPC5 Q9UL62 1/20 0.43
ITGB3 P05106 12/20 0.42
ITGAV P06756 8/20 0.42
ITGA2B P08514 5/20 0.42
ITGB1 P05556 1/20 0.40
ITGA5 P08648 1/20 0.40
CHRM2 P08172 1/20 0.40
SLC6A4 P31645 1/20 0.40
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
SPHK2 Q9NRA0 1/20 0.39
SPHK1 Q9NYA1 1/20 0.39
PIN1 Q13526 2/20 0.38
TUBB4A P04350 2/20 0.37
TUBB P07437 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7540165 0.80 ITGB3 (0.44) ITGB3ITGAVITGA2BCHRM2SLC6A4
SCHEMBL7539260 0.79 ITGB1 (0.45) BCHEITGB3ITGAVITGA2BITGB1
SCHEMBL6495002 0.78 ITGB3 (0.41) BCHETRPC3TRPC4TRPC5ITGB3
SCHEMBL7163734 0.71 ITGB3 (0.43) ITGB3ITGAVITGA2BNPC1ALDH1A1
SCHEMBL7370460 0.71 ITGB3 (0.43) ITGB3ITGAVITGA2BNPC1ALDH1A1
SCHEMBL6032775 0.69 ITGB3 (0.64) ITGB3ITGAVITGA2BCHRM2SLC6A4
SCHEMBL6505393 0.68 ITGB3 (0.42) BCHETRPC3TRPC4TRPC5ITGB3
SCHEMBL6504314 0.68 ITGB3 (0.44) BCHETRPC3TRPC4TRPC5ITGB3
SCHEMBL7329079 0.66 DAGLA (0.44) ITGB3ITGAVITGA2BCHRM2SLC6A4
SCHEMBL6503005 0.66 ITGB3 (0.51) ITGB3ITGAVITGA2BITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1208088-A2 FLUORENE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GmbH (DE) 2002-05-29 EP disclosed
WO-2001010841-A2 FLUORENE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2001-02-15 WO disclosed