SCHEMBL7329978

SCHEMBL7329978

CCOC(=O)C(=O)CSc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.56
HPGD P15428 1/20 0.56
NPC1 O15118 3/20 0.53
RAB9A P51151 2/20 0.53
TP53 P04637 1/20 0.53
FFAR1 O14842 1/20 0.53
L3MBTL1 Q9Y468 3/20 0.52
MAPK1 P28482 1/20 0.52
HSD17B10 Q99714 2/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
TSHR P16473 1/20 0.48
TDP1 Q9NUW8 1/20 0.47
MAPT P10636 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
GAA P10253 1/20 0.46
PKM P14618 1/20 0.46
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11434557 0.91 ALDH1A1 (0.48) ALDH1A1HPGDNPC1RAB9ATP53
SCHEMBL2027600 0.82 LMNA (0.59) ALDH1A1HPGDNPC1RAB9AFFAR1
SCHEMBL1326178 0.82 LMNA (0.44) ALDH1A1NPC1MEN1KMT2ATDP1
SCHEMBL20022958 0.81 FFAR1 (0.52) ALDH1A1FFAR1L3MBTL1MAPK1MEN1
SCHEMBL1324549 0.81 MTNR1B (0.51) ALDH1A1L3MBTL1MAPK1TSHRTDP1
SCHEMBL6785504 0.80 DNTT (0.43) ALDH1A1HPGDNPC1RAB9AL3MBTL1
SCHEMBL8635941 0.78 FFAR1 (0.61) ALDH1A1HPGDNPC1RAB9ATP53
SCHEMBL7513150 0.77 ALDH1A1 (0.54) ALDH1A1HPGDNPC1RAB9ATP53
SCHEMBL6421307 0.77 ALDH1A1 (0.54) ALDH1A1HPGDNPC1RAB9AFFAR1
SCHEMBL1326176 0.76 GLA (0.44) ALDH1A1HPGDNPC1RAB9ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4472380-A CARBOXYALKYL DIPEPTIDE DERIVATIVES MERCK & CO., INC. (US) 1984-09-18 US disclosed
US-4374829-A Aminoacid derivatives as antihypertensives MERCK & CO., INC. (US) 1983-02-22 US disclosed
EP-0012401-A1 Carboxyalkyl dipeptide derivatives, process for preparing them and pharmaceutical composition containing them MERCK & CO. INC. (US) 1980-06-25 EP disclosed