SCHEMBL7330358

SCHEMBL7330358

C#CC1(OCc2ccc(Cl)cc2F)CCN(C(C)=O)CC1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
RAB9A P51151 1/20 0.41
OPRL1 P41146 1/20 0.40
RORC P51449 6/20 0.37
MMP1 P03956 2/20 0.37
ADAM17 P78536 1/20 0.37
GPR183 P32249 1/20 0.37
DPP4 P27487 1/20 0.36
DPP7 Q9UHL4 1/20 0.36
FFAR4 Q5NUL3 1/20 0.36
CCR3 P51677 1/20 0.36
HPD P32754 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7324875 0.84 DPP4 (0.49) ALDH1A1MEN1KMT2ARAB9ARORC
SCHEMBL7330260 0.84 RAB9A (0.57) ALDH1A1MEN1KMT2ARAB9ADPP4
SCHEMBL11128101 0.83 RAB9A (0.56) ALDH1A1MEN1KMT2ARAB9ADPP4
SCHEMBL11128097 0.82 RAB9A (0.55) ALDH1A1MEN1KMT2ARAB9ADPP4
Oxalic Acid SCHEMBL7325487 0.70 KMT2A (0.43) ALDH1A1MEN1KMT2ARAB9ADPP4
SCHEMBL7330601 0.69 FFAR4 (0.41) MMP1ADAM17FFAR4HPD
SCHEMBL7331567 0.68 FFAR4 (0.37) ALDH1A1MMP1ADAM17GPR183FFAR4
SCHEMBL13034127 0.67 GAA (0.47) ALDH1A1HPD
SCHEMBL3088869 0.67 ALDH1A1 (0.50) ALDH1A1MEN1KMT2AOPRL1
SCHEMBL10555660 0.65 CYP2D6 (0.39) ALDH1A1RORCDPP4DPP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0102034-B1 SPIRO(2H-1,4-BENZODIOXEPIN-3(5H)4'-PIPERIDINE AND 3'-PYRROLIDINO) COMPOUNDS, A PROCESS FOR PREPARING THE SAME AND THEIR USE AS MEDICAMENTS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1988-04-20 EP disclosed
US-4521537-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1985-06-04 US disclosed
EP-0102034-A1 Spiro(2H-1,4-benzodioxepin-3(5H)4'-piperidine and 3'-pyrrolidino) compounds, a process for preparing the same and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1984-03-07 EP disclosed