SCHEMBL7330788

SCHEMBL7330788

Cc1ccc2c(c1)sc1ncc(C(O)CCc3ccccc3)n12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
KMT2A Q03164 2/20 0.42
PARP10 Q53GL7 5/20 0.41
PARP2 Q9UGN5 4/20 0.41
PARP15 Q460N3 2/20 0.41
PARP14 Q460N5 2/20 0.41
TNKS2 Q9H2K2 2/20 0.41
TNKS O95271 1/20 0.41
PARP1 P09874 1/20 0.41
TIPARP Q7Z3E1 1/20 0.41
PARP16 Q8N5Y8 1/20 0.41
PARP12 Q9H0J9 1/20 0.41
PARP11 Q9NR21 1/20 0.41
PARP4 Q9UKK3 1/20 0.41
PARP3 Q9Y6F1 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 4/20 0.37
TP53 P04637 1/20 0.37
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7332741 0.87 MAPK14 (0.37) NPC1KDM4EMAPTTP53
SCHEMBL7331144 0.86 PTPN11 (0.50) RAB9AKMT2APARP10PARP2PARP15
SCHEMBL7337608 0.86 RAB9A (0.43) NPC1RAB9AKDM4EMAPTTP53
SCHEMBL7335512 0.79 DCTPP1 (0.43) NPC1RAB9AKDM4ELMNASMN1; SMN2
SCHEMBL7330585 0.74 ALDH1A1 (0.53) NPC1RAB9AKDM4EMAPTPOLB
SCHEMBL7338080 0.73 DCTPP1 (0.42) NPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL7331138 0.71 PARP10 (0.51) NPC1RAB9AKMT2APARP10PARP2
SCHEMBL18747058 0.71 PARP10 (0.51) NPC1RAB9AKMT2APARP10PARP2
SCHEMBL7338395 0.70 DCTPP1 (0.42) NPC1RAB9AKMT2AKDM4EMAPT
SCHEMBL7329929 0.70 DCTPP1 (0.40) NPC1RAB9AKMT2AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6191124-B1 VIRICIDES PHARMACIA & UPJOHN COMPANY 2001-02-20 US claimed
EP-0757692-A1 METHANOL DERIVATIVES FOR TREATMENT OF RETROVIRAL INFECTIONS ESPECIALLY HIV INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1997-02-12 EP claimed
WO-1995029922-A1 METHANOL DERIVATIVES FOR TREATMENT OF RETROVIRAL INFECTIONS ESPECIALLY HIV INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-09 WO claimed
US-6191124-B1 VIRICIDES PHARMACIA & UPJOHN COMPANY 2001-02-20 US disclosed
EP-0757692-A1 METHANOL DERIVATIVES FOR TREATMENT OF RETROVIRAL INFECTIONS ESPECIALLY HIV INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1997-02-12 EP disclosed
WO-1995029922-A1 METHANOL DERIVATIVES FOR TREATMENT OF RETROVIRAL INFECTIONS ESPECIALLY HIV INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-09 WO disclosed