SCHEMBL7332002

SCHEMBL7332002

COc1ccc(Cl)cc1NC(=O)C1CCc2c(ncn2OC(=O)/C=C/C(=O)On2cnc3c2CCC(C(=O)Nc2cc(Cl)ccc2OC)C3)C1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C19 P33261 1/20 0.47
RBP4 P02753 1/20 0.45
MAPT P10636 2/20 0.44
NPC1 O15118 1/20 0.43
LMNA P02545 2/20 0.43
STAT3 P40763 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7330529 0.87 KDM4E (0.48) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL7324003 0.79 KDM4E (0.50) ALDH1A1CYP3A4CYP2C19MAPTLMNA
SCHEMBL7331892 0.79 TSHR (0.49) LMNAMEN1KMT2A
SCHEMBL7334780 0.78 MEN1 (0.40) ALDH1A1MAPTNPC1LMNAMEN1
SCHEMBL7334149 0.77 PTGDR2 (0.44) ALDH1A1MAPTMEN1KMT2A
SCHEMBL7325586 0.77 GAA (0.53) ALDH1A1LMNAMEN1KMT2A
SCHEMBL7335424 0.77 KMT2A (0.42) ALDH1A1MAPTNPC1LMNAMEN1
Fumaric Acid SCHEMBL7326007 0.74 ALDH1A1 (0.45) ALDH1A1CYP1A2CYP3A4CYP2C19RBP4
SCHEMBL7333021 0.73 GPBAR1 (0.34) ALDH1A1LMNAMEN1KMT2A
Fumaric Acid SCHEMBL7326008 0.73 ALDH1A1 (0.45) ALDH1A1CYP1A2CYP3A4CYP2C19RBP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0376624-B1 4,5,6,7-Tetrahydrobenzimidazole derivatives and their preparation YAMANOUCHI PHARMA CO LTD (JP) 1994-09-14 EP disclosed