SCHEMBL7332157

SCHEMBL7332157

CCN1CCN(c2cc(-c3ccc(F)cc3)c3c(n2)C2CCC(C3)C2)CC1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.57
HTR2A P28223 5/20 0.57
HRH4 Q9H3N8 1/20 0.40
HTT P42858 2/20 0.36
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 3/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
KDM2B Q8NHM5 1/20 0.35
SCN9A Q15858 1/20 0.35
MAPT P10636 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
CSNK1D P48730 1/20 0.34
MAPK11 Q15759 1/20 0.34
MAPK14 Q16539 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9788682 0.84 DRD2 (0.57) DRD2HTR2AHRH4HTTKDM4E
SCHEMBL7327599 0.83 DRD2 (0.55) DRD2HTR2AHRH4HTTKDM4E
SCHEMBL9614388 0.75 DRD2 (0.70) DRD2HTR2AHRH4HTTKDM4E
SCHEMBL7425400 0.73 DRD2 (0.44) DRD2HTR2AKDM4EALDH1A1SMN1; SMN2
SCHEMBL7329861 0.73 DRD2 (0.44) DRD2HTR2AHTTKDM4EALDH1A1
SCHEMBL7333157 0.73 DRD2 (0.93) DRD2HTR2AHRH4HTTKDM4E
SCHEMBL7334897 0.72 DRD2 (1.00) DRD2HTR2AHRH4HTTKDM4E
Blonanserin SCHEMBL29379647 0.72 DRD2 (1.00) DRD2HTR2AHRH4HTTKDM4E
Blonanserin SCHEMBL119669 0.72 DRD2 (1.00) DRD2HTR2AHRH4HTTKDM4E
SCHEMBL9440217 0.72 DRD2 (0.63) DRD2HTR2AHRH4HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0385237-B1 2-(1-piperazinyl)-4-phenylcycloalkanopyridine derivatives, processes for the production thereof, and pharmaceutical composition containing the same DAINIPPON PHARMACEUTICAL CO (JP) 1994-06-29 EP disclosed
US-5021421-A Psychotropic agents DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1991-06-04 US disclosed
EP-0385237-A2 2-(1-piperazinyl)-4-phenylcycloalkanopyridine derivatives, processes for the production thereof, and pharmaceutical composition containing the same DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1990-09-05 EP disclosed