SCHEMBL7332296

SCHEMBL7332296

CC(C)[C@H](NC(=O)[C@H](C)NC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)OCc1ccccc1)C(C)C

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 4/20 0.70
REN P00797 4/20 0.61
CTSK P43235 4/20 0.54
CTSB P07858 3/20 0.54
ELANE P08246 1/20 0.52
TRPM8 Q7Z2W7 1/20 0.52
ECE1 P42892 2/20 0.52
MME P08473 1/20 0.52
PSMB11 A5LHX3 3/20 0.51
PSMA7 O14818 3/20 0.51
PSMB1 P20618 3/20 0.51
PSMA1 P25786 3/20 0.51
PSMA2 P25787 3/20 0.51
PSMA3 P25788 3/20 0.51
PSMA4 P25789 3/20 0.51
PSMB8 P28062 3/20 0.51
PSMB9 P28065 3/20 0.51
PSMA5 P28066 3/20 0.51
PSMB4 P28070 3/20 0.51
PSMB6 P28072 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15095633 0.98 CTSD (0.70) CTSDRENCTSKCTSBELANE
SCHEMBL6132144 0.93 CTSD (0.76) CTSDRENCTSKCTSBTRPM8
SCHEMBL6449641 0.93 CTSD (0.76) CTSDRENCTSKCTSBTRPM8
Acetic Acid SCHEMBL7270658 0.91 CTSD (0.73) CTSDRENCTSKCTSBTRPM8
SCHEMBL9232828 0.91 CTSD (0.76) CTSDRENCTSKCTSBTRPM8
SCHEMBL9740721 0.91 CTSD (0.76) CTSDRENCTSKCTSBTRPM8
SCHEMBL6446780 0.91 CTSD (0.76) CTSDRENCTSKCTSBTRPM8
SCHEMBL6446151 0.91 CTSD (0.76) CTSDRENCTSKCTSBTRPM8
SCHEMBL6445103 0.91 CTSD (0.76) CTSDRENCTSKCTSBTRPM8
SCHEMBL6446525 0.91 CTSD (0.60) CTSDRENCTSKCTSBTRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed