SCHEMBL6446525

SCHEMBL6446525

C[C@H](NC(=O)OCc1ccccc1)C(=O)NC(Cc1ccccc1)C(O)C(O)C(Cc1ccccc1)NC(=O)[C@H](C)NC(=O)OCc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSD P07339 3/20 0.60
CTSK P43235 5/20 0.59
REN P00797 2/20 0.56
TRPM8 Q7Z2W7 1/20 0.55
TACR1 P25103 2/20 0.54
CTRB1 P17538 2/20 0.53
CTSL P07711 3/20 0.53
CTSS P25774 3/20 0.53
CTSB P07858 2/20 0.53
CYP1A2 P05177 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15095633 0.93 CTSD (0.70) CTSDCTSKRENTRPM8CTSB
SCHEMBL7332296 0.91 CTSD (0.70) CTSDCTSKRENTRPM8CTSB
SCHEMBL4949767 0.88 TRPM8 (0.64) CTSDCTSKTRPM8TACR1CTRB1
SCHEMBL2736202 0.88 TRPM8 (0.64) CTSDCTSKTRPM8TACR1CTRB1
SCHEMBL7337287 0.88 TRPM8 (0.64) CTSDCTSKTRPM8TACR1CTRB1
SCHEMBL2736218 0.88 TRPM8 (0.64) CTSDCTSKTRPM8TACR1CTRB1
SCHEMBL9421829 0.88 TRPM8 (0.64) CTSDCTSKTRPM8TACR1CTRB1
SCHEMBL5916913 0.88 TRPM8 (0.64) CTSDCTSKTRPM8TACR1CTRB1
SCHEMBL6446780 0.88 CTSD (0.76) CTSDCTSKRENTRPM8TACR1
SCHEMBL6446151 0.88 CTSD (0.76) CTSDCTSKRENTRPM8TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-B1 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LAB (US) 2005-08-17 EP disclosed
EP-0402646-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 1998-07-22 EP disclosed
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed