SCHEMBL7333301

SCHEMBL7333301

COc1ccc(-c2ccc3[nH]cc(CC#N)c3c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 2/20 0.56
GPR84 Q9NQS5 2/20 0.55
HTR2B P41595 3/20 0.52
HTR2A P28223 6/20 0.50
HTR1A P08908 4/20 0.50
HTR2C P28335 3/20 0.50
CYP2D6 P10635 2/20 0.50
CYP1A2 P05177 2/20 0.50
HTR1D P28221 2/20 0.50
HTR1B P28222 2/20 0.50
HTR7 P34969 2/20 0.50
HTR6 P50406 2/20 0.50
HTR4 Q13639 2/20 0.50
MAPT P10636 1/20 0.50
TSHR P16473 1/20 0.50
NFKB1 P19838 1/20 0.50
TRPM8 Q7Z2W7 1/20 0.50
BLM P54132 1/20 0.49
PMP22 Q01453 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2724551 0.89 GPR84 (0.69) CSNK2A1GPR84HTR2BHTR2AHTR1A
SCHEMBL8868480 0.86 GPR84 (0.58) CSNK2A1GPR84HTR2BHTR2AHTR1A
SCHEMBL6574193 0.83 CSNK2A1 (0.61) CSNK2A1SLC6A4
SCHEMBL7335081 0.82 CSNK2A1 (0.60) CSNK2A1GPR84HTR2AMAPTTRPM8
SCHEMBL7327065 0.82 CSNK2A1 (0.60) CSNK2A1GPR84HTR2AHTR1ATSHR
SCHEMBL2727889 0.80 HTR2A (0.62) CSNK2A1GPR84HTR2BHTR2AHTR1A
SCHEMBL7331404 0.80 HTR1A (0.79) HTR2BHTR2AHTR1AHTR2CCYP2D6
SCHEMBL4945471 0.78 CSNK2A1 (0.56) CSNK2A1GPR84HTR1DHTR1BSLC6A4
SCHEMBL7332860 0.77 HTR1D (0.80) HTR2BHTR2AHTR1AHTR2CCYP2D6
SCHEMBL18311441 0.77 HTR1B (0.56) CSNK2A1GPR84HTR2BHTR2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0674620-A1 TRYPTAMINE ANALOGUES AS 5-HT 1?-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-10-04 EP disclosed
WO-1994014771-A1 TRYPTAMINE ANALOGUES AS 5-HT1-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-07-07 WO disclosed