SCHEMBL7334206

SCHEMBL7334206

CC(C)[C@H](NC(=O)N(C)CCc1ccccn1)C(=O)Oc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.47
RAB9A P51151 3/20 0.47
MEN1 O00255 2/20 0.47
NPC1 O15118 1/20 0.47
POLB P06746 1/20 0.47
HIF1A Q16665 1/20 0.44
CA2 P00918 2/20 0.42
ALDH1A1 P00352 4/20 0.42
KDM4E B2RXH2 3/20 0.42
L3MBTL1 Q9Y468 1/20 0.40
TDP1 Q9NUW8 2/20 0.40
HSD11B1 P28845 1/20 0.40
LMNA P02545 2/20 0.39
MITF O75030 1/20 0.39
GAA P10253 1/20 0.39
AGTR1 P30556 1/20 0.39
OPRK1 P41145 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4680500 0.92 CA2 (0.51) KMT2ARAB9AMEN1NPC1POLB
SCHEMBL4680503 0.92 CA2 (0.51) KMT2ARAB9AMEN1NPC1POLB
SCHEMBL4679453 0.85 CA2 (0.46) KMT2ARAB9AMEN1NPC1POLB
SCHEMBL4679457 0.85 CA2 (0.46) KMT2ARAB9AMEN1NPC1POLB
SCHEMBL7311190 0.84 TRPM8 (0.45) KMT2ARAB9AMEN1NPC1CA2
SCHEMBL7333765 0.84 ALDH1A1 (0.44) KMT2ARAB9AMEN1NPC1POLB
SCHEMBL7311193 0.84 TRPM8 (0.45) KMT2ARAB9AMEN1NPC1CA2
SCHEMBL4679034 0.82 KMT2A (0.48) KMT2ARAB9AMEN1NPC1ALDH1A1
SCHEMBL4679037 0.82 KMT2A (0.48) KMT2ARAB9AMEN1NPC1ALDH1A1
SCHEMBL7334203 0.80 ALDH1A1 (0.41) KMT2ARAB9AMEN1NPC1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed