SCHEMBL7334559

SCHEMBL7334559

Cc1cc(O)cc(N2C(=O)c3ccccc3C2=O)c1

nearest known ligand 0.77

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 6/20 0.58
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
ESR1 P03372 3/20 0.51
NR1H3 Q13133 2/20 0.49
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
PIM3 Q86V86 1/20 0.46
HIPK4 Q8NE63 1/20 0.46
SCN2A Q99250 1/20 0.46
ESR2 Q92731 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30792888 0.87 GRM5 (0.62) GRM5MEN1KMT2ANPC1RAB9A
SCHEMBL5604859 0.87 GRM5 (0.62) GRM5MEN1KMT2ANPC1RAB9A
SCHEMBL7386922 0.81 GRM5 (0.56) GRM5MEN1KMT2A
SCHEMBL12034643 0.81 ESR1 (0.46) GRM5MEN1KMT2AESR1NPC1
SCHEMBL20437115 0.79 LMNA (0.44) GRM5ESR1NPC1RAB9AESR2
SCHEMBL12034645 0.77 CA9 (0.48) ESR1ESR2
SCHEMBL1662738 0.77 ESR1 (0.80) GRM5MEN1KMT2AESR1NR1H3
SCHEMBL30758580 0.77 MEN1 (0.67) MEN1KMT2ANR1H3SCN2A
SCHEMBL30777591 0.77 MEN1 (0.67) MEN1KMT2ANR1H3SCN2A
SCHEMBL259386 0.77 MEN1 (0.67) MEN1KMT2ANR1H3SCN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0778839-B1 NOVEL PHOSPHANE OXIDES, METHOD OF PREPARING THEM AND DRUGS CONTAINING THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1998-12-23 EP disclosed
EP-0687253-B1 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME BOEHRINGER MANNHEIM GMBH (DE) 1998-12-16 EP disclosed
US-5824679-A Phosphanoxides--preparation and use BOEHRINGER MANNHEIM GMBH (DE) 1998-10-20 US disclosed
US-5795892-A ANTICOAGULANTS BOEHRINGER MANNEIM GMBH (DE) 1998-08-18 US disclosed
EP-0778829-A1 NOVEL 4-AMINOPYRIDAZINES, METHOD OF PREPARING THEM AND DRUGS CONTAINING THESE COMPOUNDS Roche Diagnostics GmbH (DE) 1997-06-18 EP disclosed
WO-1996006832-A1 NOVEL 4-AMINOPYRIDAZINES, METHOD OF PREPARING THEM AND DRUGS CONTAINING THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1996-03-07 WO disclosed
EP-0687253-A1 NEW 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME Roche Diagnostics GmbH (DE) 1995-12-20 EP disclosed
WO-1994020467-A1 NEW 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME BOEHRINGER MANNHEIM GMBH (DE) 1994-09-15 WO disclosed