SCHEMBL7335403

SCHEMBL7335403

Cc1cc(C2=NNC(=O)CC2C(C)C)ccc1[O]

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 6/20 0.56
PDE3B Q13370 12/20 0.44
PDE3A Q14432 12/20 0.44
PDE4A P27815 2/20 0.42
PDE4B Q07343 2/20 0.42
PDE4C Q08493 2/20 0.42
PDE4D Q08499 2/20 0.42
GALR3 O60755 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7299065 0.86 PDE3B (0.55) GPR119PDE3BPDE3APDE4APDE4B
SCHEMBL9686166 0.86 GPR119 (0.55) GPR119PDE3BPDE3APDE4APDE4B
SCHEMBL9688044 0.82 PDE3B (0.64) GPR119PDE3BPDE3APDE4APDE4B
SCHEMBL9687496 0.82 GPR119 (0.53) GPR119PDE3BPDE3APDE4APDE4B
SCHEMBL7296587 0.80 GPR119 (0.57) GPR119PDE3BPDE3APDE4APDE4B
SCHEMBL9686551 0.79 GPR119 (0.56) GPR119PDE3BPDE3A
SCHEMBL9686159 0.78 GPR119 (0.64) GPR119
SCHEMBL9687501 0.78 GPR119 (0.52) GPR119PDE3BPDE3APDE4APDE4B
SCHEMBL7332519 0.78 GPR119 (0.50) GPR119PDE3BPDE3APDE4APDE4B
SCHEMBL7298045 0.77 GPR119 (0.63) GPR119PDE3BPDE3APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135932-A 2-HYDROXYPROPYLAMINO-ALKYL-BENZIMIDAZOLY-5-YL DERIVATIVES AND THEIR USE IN THE TREATMENT OF HEART DISEASE DR. KARL THOMAE GMBH (DE) 1992-08-04 US disclosed
EP-0400519-A1 2-Hydroxy-n-propylamines, medicaments containing these compounds and method for preparing them Dr. Karl Thomae GmbH (DE) 1990-12-05 EP disclosed