SCHEMBL7335803

SCHEMBL7335803

CC(C)(C)OC(=O)N1CCC(Oc2ccc(CBr)c(OC(F)(F)F)c2)CC1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 6/20 0.52
EPHX2 P34913 2/20 0.46
OXTR P30559 1/20 0.46
PDE4D Q08499 3/20 0.46
PDE4A P27815 2/20 0.46
PDE4B Q07343 2/20 0.46
PDE4C Q08493 2/20 0.46
LIPE Q05469 1/20 0.46
HRH3 Q9Y5N1 1/20 0.45
ALDH1A1 P00352 1/20 0.43
CHEK2 O96017 1/20 0.43
NEK2 P51955 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7335892 0.91 GPR119 (0.56) GPR119EPHX2OXTRPDE4DPDE4A
SCHEMBL7337034 0.89 GPR119 (0.52) GPR119EPHX2OXTRPDE4DPDE4A
SCHEMBL7339211 0.87 GPR119 (0.54) GPR119EPHX2OXTRPDE4DPDE4A
SCHEMBL8088539 0.86 EPHX2 (0.60) GPR119EPHX2PDE4DPDE4APDE4B
SCHEMBL7343837 0.85 GPR119 (0.48) GPR119EPHX2OXTRPDE4DPDE4A
SCHEMBL2951108 0.81 GPR119 (0.63) GPR119EPHX2LIPEHRH3ALDH1A1
SCHEMBL8088551 0.79 EPHX2 (0.62) GPR119EPHX2PDE4DPDE4APDE4B
SCHEMBL3344947 0.78 GPR119 (0.61) GPR119PDE4DPDE4APDE4BPDE4C
SCHEMBL7333649 0.78 GPR119 (0.50) GPR119EPHX2OXTRPDE4DPDE4A
SCHEMBL23410126 0.78 GPR119 (0.58) GPR119EPHX2PDE4BLIPEHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090805-A Tocolytic oxytocin receptor antagonists MERCK & CO., INC. (US) 2000-07-18 US disclosed
US-5968938-A Piperazine oxytocin receptor antagonists MERCK & CO., INC. (US) 1999-10-19 US disclosed