SCHEMBL7336189

SCHEMBL7336189

COc1cc(C(=O)N(C)c2ccccc2C)ccc1NC(=O)c1ccccc1OC(C)=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
MAPT P10636 6/20 0.49
RAB9A P51151 5/20 0.49
NPC1 O15118 2/20 0.49
GAA P10253 2/20 0.47
TP53 P04637 1/20 0.47
BRPF1 P55201 2/20 0.45
BRD4 O60885 1/20 0.45
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.45
POLB P06746 2/20 0.43
KCNMA1 Q12791 1/20 0.43
KCNK3 O14649 1/20 0.43
KCNK9 Q9NPC2 1/20 0.43
TDP1 Q9NUW8 2/20 0.43
TOP1 P11387 1/20 0.43
ABL1 P00519 1/20 0.43
RIN1 Q13671 1/20 0.43
IRAK4 Q9NWZ3 1/20 0.43
PKM P14618 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7345983 0.87 MAPT (0.58) ALDH1A1MAPTRAB9ANPC1GAA
Hydrochloric Acid SCHEMBL7336895 0.83 ALDH1A1 (0.45) ALDH1A1MAPTRAB9ANPC1GAA
SCHEMBL7378000 0.83 ALDH1A1 (0.51) ALDH1A1MAPTRAB9ANPC1GAA
SCHEMBL7340419 0.82 TP53 (0.51) ALDH1A1MAPTRAB9ANPC1GAA
SCHEMBL7344448 0.81 PYGL (0.58) ALDH1A1MAPTRAB9ANPC1GAA
SCHEMBL8636243 0.79 BRD4 (0.49) ALDH1A1RAB9ANPC1GAATP53
SCHEMBL7342516 0.79 ALDH1A1 (0.41) ALDH1A1MAPTRAB9ANPC1GAA
SCHEMBL7345419 0.78 TP53 (0.44) ALDH1A1MAPTRAB9ANPC1GAA
SCHEMBL7337480 0.78 TP53 (0.42) ALDH1A1MAPTRAB9ANPC1GAA
SCHEMBL7427909 0.77 TP53 (0.43) ALDH1A1MAPTRAB9ANPC1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832061-B1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 2001-09-05 EP disclosed
US-6054457-A Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-25 US disclosed
WO-1996041795-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-12-27 WO disclosed