SCHEMBL7336336

SCHEMBL7336336

CC(C)[C@H](NC(=O)OCc1ccccn1)C(=O)N[C@@H](Cc1ccccc1)[C@H](O)[C@H](O)[C@H](Cc1ccccc1)NC(=O)OCc1cccnc1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.60
CTSD P07339 4/20 0.55
CYP3A4 P08684 4/20 0.49
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C19 P33261 1/20 0.45
CASP3 P42574 1/20 0.44
CASP7 P55210 1/20 0.44
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
REN P00797 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7334719 1.00 CA2 (0.60) CA2CTSDCYP3A4CYP1A2CYP2D6
SCHEMBL7334173 1.00 CA2 (0.60) CA2CTSDCYP3A4CYP1A2CYP2D6
SCHEMBL7332791 1.00 CA2 (0.60) CA2CTSDCYP3A4CYP1A2CYP2D6
SCHEMBL6448343 0.92 CTSD (0.63) CA2CTSDCYP3A4CYP1A2CYP2D6
SCHEMBL6447680 0.92 CA2 (0.69) CA2CTSDCYP1A2CYP2D6CASP3
SCHEMBL6445023 0.92 CA2 (0.69) CA2CTSDCYP1A2CYP2D6CASP3
SCHEMBL7343161 0.92 CA2 (0.69) CA2CTSDCYP1A2CYP2D6CASP3
SCHEMBL6446319 0.92 CTSD (0.63) CA2CTSDCYP3A4CYP1A2CYP2D6
SCHEMBL9227910 0.92 CA2 (0.69) CA2CTSDCYP1A2CYP2D6CASP3
SCHEMBL6449063 0.92 CA2 (0.69) CA2CTSDCYP1A2CYP2D6CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed