SCHEMBL7336907

SCHEMBL7336907

CCOC(=O)CCCN(c1ccccc1C(=O)OC)S(=O)(=O)c1ccccc1C

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 1/20 0.43
KMT2A Q03164 1/20 0.42
HSD17B10 Q99714 2/20 0.40
USP2 O75604 1/20 0.40
MAPT P10636 2/20 0.40
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
ALOX5 P09917 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA5A P35218 1/20 0.39
CA9 Q16790 1/20 0.39
PTGER1 P34995 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
POLB P06746 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8653909 0.94 HCRTR2 (0.44) HCRTR2KMT2AHSD17B10USP2MAPT
SCHEMBL1495969 0.85 TP53 (0.52) KMT2AMAPTALDH1A1PTGER1L3MBTL1
SCHEMBL4867236 0.82 LMNA (0.41) HCRTR2KMT2AHSD17B10MAPTKDM4E
SCHEMBL14408832 0.72 TSHR (0.54) HSD17B10USP2KDM4EALDH1A1ALOX5
SCHEMBL25333728 0.72 PSEN1 (0.43) HCRTR2KMT2AMAPTL3MBTL1POLB
SCHEMBL23209700 0.72 MMP1 (0.46) HCRTR2MAPTALDH1A1PTGER1L3MBTL1
SCHEMBL1291299 0.72 PSEN1 (0.51) HCRTR2MAPTL3MBTL1TP53
SCHEMBL28331917 0.69 CA12 (0.49) HSD17B10USP2ALDH1A1CA9
SCHEMBL6541841 0.69 L3MBTL1 (0.63) ALOX5CA1CA2CA5ACA9
SCHEMBL9037934 0.68 KMT2A (0.51) KMT2AHSD17B10MAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022282-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1996-07-25 WO disclosed