SCHEMBL7337019

SCHEMBL7337019

N#Cc1ccc2cc(/C=C/c3ccc(C(N)=O)cc3)ccc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 2/20 0.53
PARP15 Q460N3 1/20 0.53
PARP2 Q9UGN5 1/20 0.53
PLG P00747 2/20 0.46
PLAU P00749 2/20 0.46
PLAT P00750 1/20 0.46
KLK1 P06870 1/20 0.46
P4HB P07237 8/20 0.45
MAPT P10636 2/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
F2 P00734 1/20 0.42
KLKB1 P03952 1/20 0.42
PRSS1 P07477 1/20 0.42
MYC P01106 3/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
CYP3A4 P08684 1/20 0.40
HDAC2 Q92769 1/20 0.40
PARP3 Q9Y6F1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7337024 1.00 PARP10 (0.53) PARP10PARP15PARP2PLGPLAU
SCHEMBL7341383 0.87 MAPT (0.47) PLGPLAUPLATKLK1P4HB
SCHEMBL7341392 0.87 MAPT (0.47) PLGPLAUPLATKLK1P4HB
SCHEMBL23909542 0.82 PARP15 (0.59) PARP10PARP15PARP2PLGPLAU
SCHEMBL10068047 0.79 RELA (0.52) PLGPLAUPLATKLK1P4HB
SCHEMBL7338903 0.78 RELA (0.63) PLGPLAUPLATKLK1MAPT
SCHEMBL6635557 0.78 LCK (0.55) PARP10PARP15PARP2PLGPLAU
SCHEMBL7338887 0.78 RELA (0.63) PLGPLAUPLATKLK1MAPT
SCHEMBL27536270 0.77 PLAU (0.74) PLGPLAUPLATKLK1MAPT
SCHEMBL7345218 0.77 CA1 (0.53) P4HBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20010049374-A1 Urokinase inhibitors STEELE ANDREW W (US) 2001-12-06 US disclosed
US-6284796-B1 NAPHTHAMIDINE COMPOUNDS ABBOTT LABORATORIES 2001-09-04 US disclosed
US-6258822-B1 ENZYME INHIBITORS OF NAPHTHALENE AMIDINE COMPOUNDS ABBOTT LABORATORIES 2001-07-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010049374-A1 Urokinase inhibitors SERPINE1, PLAU, SERPINB1 PARP10 1727/4885PARP15 1589/4885PARP2 2515/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.