SCHEMBL7337442

SCHEMBL7337442

N[C@@H](Cc1ccccc1)[C@@H](O)C(F)(F)[C@@H](N)Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.49
LMNA P02545 1/20 0.49
MAPK1 P28482 1/20 0.49
SLC15A1 P46059 1/20 0.44
EPHX1 P07099 1/20 0.44
CSNK1E P49674 1/20 0.43
ALPI P09923 1/20 0.42
PKM P14618 1/20 0.42
PTGS1 P23219 1/20 0.42
XIAP P98170 1/20 0.42
SLC7A5 Q01650 1/20 0.42
SLC6A2 P23975 2/20 0.41
TAAR1 Q96RJ0 2/20 0.41
MAOA P21397 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
CYP2A6 P11509 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275924 1.00 KDM4E (0.49) KDM4ELMNAMAPK1SLC15A1EPHX1
SCHEMBL10622532 0.84 EPHX1 (0.48) KDM4ELMNAMAPK1SLC15A1EPHX1
SCHEMBL6556276 0.84 EPHX1 (0.48) KDM4ELMNAMAPK1SLC15A1EPHX1
Hydrochloric Acid SCHEMBL5711578 0.82 EPHX1 (0.47) KDM4ELMNAMAPK1SLC15A1EPHX1
SCHEMBL10432270 0.80 ALPI (0.47) SLC15A1CSNK1EALPIPKMPTGS1
SCHEMBL27345872 0.79 SLC15A1 (0.44) KDM4ELMNAMAPK1SLC15A1EPHX1
SCHEMBL10445629 0.79 MDM2 (0.49) SLC15A1EPHX1CSNK1EALPIPKM
SCHEMBL7412831 0.78 SLC15A1 (0.50) SLC15A1EPHX1CSNK1EALPIPKM
SCHEMBL6351074 0.78 SLC15A1 (0.43) KDM4ELMNAMAPK1SLC15A1EPHX1
SCHEMBL7412834 0.78 SLC15A1 (0.50) SLC15A1EPHX1CSNK1EALPIPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed