SCHEMBL7338378

SCHEMBL7338378

N#CCc1cccc(Cl)c1OCC(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 1/20 0.36
CACNG8 Q8WXS5 1/20 0.36
ALDH1A1 P00352 3/20 0.33
RECQL P46063 1/20 0.33
MRGPRX4 Q96LA9 2/20 0.33
SLC22A12 Q96S37 1/20 0.33
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2C19 P33261 2/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
ALOX12 P18054 1/20 0.32
AR P10275 2/20 0.32
HPGD P15428 2/20 0.32
KDM4E B2RXH2 2/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14956297 0.80 KMT2A (0.47) ALDH1A1RECQLMRGPRX4KMT2AMEN1
SCHEMBL7334130 0.80 KMT2A (0.35) ALDH1A1RECQLMRGPRX4KMT2AMEN1
SCHEMBL3531950 0.76 GRIA1 (0.40) GRIA1CACNG8ALDH1A1KMT2AMEN1
SCHEMBL16822093 0.76 GRIA1 (0.40) GRIA1CACNG8ALDH1A1KMT2AMEN1
SCHEMBL7344131 0.75 FABP4 (0.53) KMT2A
SCHEMBL26162784 0.72 KMT2A (0.37) ALDH1A1RECQLKMT2AMEN1CYP1A2
SCHEMBL7341969 0.72 KDM4E (0.51) KMT2ACYP1A2CYP2C19CYP3A4CYP2D6
SCHEMBL10532535 0.72 ALDH1A1 (0.43) ALDH1A1RECQLMRGPRX4KMT2AMEN1
Hydrochloric Acid SCHEMBL10533956 0.71 ALDH1A1 (0.42) ALDH1A1RECQLMRGPRX4KMT2AMEN1
SCHEMBL2744577 0.70 GRIA1 (0.42) GRIA1CACNG8ALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090805-A Tocolytic oxytocin receptor antagonists MERCK & CO., INC. (US) 2000-07-18 US disclosed
US-5968938-A Piperazine oxytocin receptor antagonists MERCK & CO., INC. (US) 1999-10-19 US disclosed