SCHEMBL7338656

SCHEMBL7338656

N=C(N)c1cc2c([nH]c1=O)CCc1cnccc1-2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 5/20 0.36
CYP11B1 P15538 4/20 0.36
CYP19A1 P11511 3/20 0.36
CDC7 O00311 3/20 0.36
DAO P14920 2/20 0.34
PKN2 Q16513 3/20 0.34
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ROCK2 O75116 3/20 0.32
AAK1 Q2M2I8 1/20 0.32
PKN1 Q16512 2/20 0.32
CDK8 P49336 2/20 0.32
PLK4 O00444 1/20 0.32
MAPK13 O15264 1/20 0.32
DAPK3 O43293 1/20 0.32
DYRK3 O43781 1/20 0.32
RPS6KA5 O75582 1/20 0.32
RPS6KA4 O75676 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7346574 0.93 KDM4E (0.39) CYP11B2CYP11B1CYP19A1CDC7DAO
SCHEMBL7341653 0.82 PKN2 (0.32) CYP11B2CYP11B1CYP19A1CDC7DAO
SCHEMBL7342355 0.81 CES1 (0.40) KDM4EALDH1A1HPGDHSD17B10TDP1
SCHEMBL7338490 0.81 AURKB (0.44) CDC7DAOPKN2KDM4EALDH1A1
SCHEMBL7347683 0.81 KDM4E (0.43) CYP11B2CDC7PKN2KDM4EALDH1A1
Hydrochloric Acid SCHEMBL7337010 0.80 CES1 (0.39) KDM4EALDH1A1HPGDHSD17B10TDP1
SCHEMBL11074795 0.79 CDC7 (0.34) CYP11B2CYP11B1CDC7PKN2
SCHEMBL7346248 0.78 SIRT3 (0.41) CYP11B2CDC7DAOKDM4EROCK2
SCHEMBL7347592 0.77 MAPK14 (0.39)
SCHEMBL7346402 0.75 KDM4E (0.48) CYP11B2CDC7KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4511569-A Tricyclic lactams and derivatives useful in increasing cardiac contractility SCHERING CORPORATION (US) 1985-04-16 US disclosed
EP-0102046-A1 Tricyclic lactams, method for making them, pharmaceutical compositions containing them SCHERING CORPORATION (US) 1984-03-07 EP disclosed