SCHEMBL7338688

SCHEMBL7338688

C/C(=N/NC(N)=S)C1CCC2(CCC(O)CC2)CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 1/20 0.61
ALDH1A1 P00352 8/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
NR2F2 P24468 1/20 0.42
ALOX12 P18054 2/20 0.40
NPSR1 Q6W5P4 3/20 0.38
CCR6 P51684 2/20 0.38
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
LMNA P02545 4/20 0.36
NPC1 O15118 1/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C19 P33261 1/20 0.35
HPGD P15428 1/20 0.33
KDM4E B2RXH2 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
ATM Q13315 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7340579 0.84 CTSK (0.41) CTSKALDH1A1MEN1KMT2ALMNA
SCHEMBL7340575 0.84 CTSK (0.41) CTSKALDH1A1MEN1KMT2ALMNA
SCHEMBL7340458 0.73 ATP1A1 (0.37)
SCHEMBL7338693 0.68 ALDH1A1 (0.44) ALDH1A1NPSR1GAAKDM4E
SCHEMBL7338613 0.66
SCHEMBL12687548 0.61
SCHEMBL844254 0.61 CTSK (0.56) CTSKALDH1A1SMN1; SMN2NR2F2ALOX12
SCHEMBL233447 0.60
SCHEMBL11937851 0.59 CTSK (0.68) CTSKALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL3209003 0.59 CTSK (0.68) CTSKALDH1A1SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0578080-B1 3,9-disubstituted-spiro (5.5)undecanes active on the cardiovascular system, process for their preparation and pharmaceutical composition containing same SIGMA TAU IND FARMACEUTI (IT) 1997-04-23 EP claimed
EP-0578080-A2 3,9-disubstituted-spiro (5.5)undecanes active on the cardiovascular system, process for their preparation and pharmaceutical composition containing same Sigma-Tau Industrie Farmaceutiche Riunite S.p.A. (IT) 1994-01-12 EP claimed
EP-0578080-B1 3,9-disubstituted-spiro (5.5)undecanes active on the cardiovascular system, process for their preparation and pharmaceutical composition containing same SIGMA TAU IND FARMACEUTI (IT) 1997-04-23 EP disclosed
US-5444082-A Treats hypertension and heart failure SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A. (IT) 1995-08-22 US disclosed
EP-0578080-A2 3,9-disubstituted-spiro (5.5)undecanes active on the cardiovascular system, process for their preparation and pharmaceutical composition containing same Sigma-Tau Industrie Farmaceutiche Riunite S.p.A. (IT) 1994-01-12 EP disclosed