SCHEMBL7339060

SCHEMBL7339060

COc1ccc(O[C@@]2(C(=O)O)CCCN2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
CTSK P43235 2/20 0.38
CES2 O00748 2/20 0.38
CES1 P23141 2/20 0.38
ALDH1A1 P00352 2/20 0.38
TET3 O43151 1/20 0.37
KMT2A Q03164 1/20 0.37
FBXL19 Q6PCT2 1/20 0.37
CXXC5 Q7LFL8 1/20 0.37
TET1 Q8NFU7 1/20 0.37
KDM2B Q8NHM5 1/20 0.37
CXXC4 Q9H2H0 1/20 0.37
KDM2A Q9Y2K7 1/20 0.37
HPGD P15428 1/20 0.37
SLC6A3 Q01959 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PARP1 P09874 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10874561 0.86 GAA (0.34) CA1CA2KMT2APARP10
SCHEMBL7341358 0.85 AKR1C1 (0.38) CTSKALDH1A1KMT2ASLC6A3
SCHEMBL7347177 0.84 HSD11B1 (0.36)
SCHEMBL10658975 0.84 HSD11B1 (0.36)
SCHEMBL7342000 0.80 HDAC3 (0.38) CTSKALDH1A1SMN1; SMN2
SCHEMBL7345830 0.78 MAPT (0.42) CES2CES1ALDH1A1KMT2AHPGD
SCHEMBL11164078 0.77 MMP14 (0.44) KMT2A
SCHEMBL15664683 0.77 TET3 (0.42) CA1CA2ALDH1A1TET3KMT2A
SCHEMBL7342381 0.76 HDAC3 (0.43) CTSKALDH1A1KMT2AHPGDCYP2C19
SCHEMBL11091264 0.74 NR4A2 (0.52) ALDH1A1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4316906-A HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1982-02-23 US disclosed