SCHEMBL7339128

SCHEMBL7339128

CCOC(=O)CCC#CNC(=O)CNC(=O)c1cccc(NCC(=NC#N)NC)c1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRK2 P25098 3/20 0.35
GRK3 P35626 3/20 0.35
KMT2A Q03164 4/20 0.34
MEN1 O00255 2/20 0.34
SMN1; SMN2 Q16637 3/20 0.33
ALDH1A1 P00352 3/20 0.33
GAA P10253 2/20 0.33
GRK5 P34947 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 2/20 0.32
TP53 P04637 1/20 0.32
GLA P06280 1/20 0.32
RAB9A P51151 1/20 0.32
GPR139 Q6DWJ6 1/20 0.32
MAPT P10636 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
TSHR P16473 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6777103 0.88 ITGB1 (0.38) KMT2AMEN1SMN1; SMN2ALDH1A1GAA
SCHEMBL7342958 0.80 KMT2A (0.41) KMT2AMEN1SMN1; SMN2ALDH1A1GAA
SCHEMBL6783445 0.79 KMT2A (0.40) KMT2AMEN1SMN1; SMN2ALDH1A1GAA
SCHEMBL7343782 0.78 ALDH1A1 (0.39) KMT2AMEN1SMN1; SMN2ALDH1A1GAA
SCHEMBL6777356 0.76 ITGB1 (0.42) SMN1; SMN2GAANPC1RAB9AGPR139
SCHEMBL6776736 0.76 NAMPT (0.48) KMT2AMEN1ALDH1A1NPC1TP53
SCHEMBL27485848 0.74 LMNA (0.48) KMT2AMEN1ALDH1A1NPC1TP53
SCHEMBL27485163 0.72 KDM4E (0.35) KMT2AMEN1SMN1; SMN2ALDH1A1GAA
SCHEMBL6776712 0.68 KDM4E (0.41) KMT2AMEN1SMN1; SMN2ALDH1A1GAA
SCHEMBL6777100 0.67 ITGB3 (0.43) KMT2AMEN1SMN1; SMN2ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP disclosed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO disclosed