SCHEMBL7339294

SCHEMBL7339294

Cc1ccc(CC(N)C(O)C(C(=O)OC(C)(C)C)C(N)c2ccccc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 1/20 0.39
LTA4H P09960 2/20 0.38
LAP3 P28838 1/20 0.37
SLC15A1 P46059 1/20 0.37
ITGA4 P13612 1/20 0.36
ITGB7 P26010 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
PKM P14618 1/20 0.36
ATM Q13315 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SLC7A5 Q01650 1/20 0.35
MAPT P10636 3/20 0.35
NPSR1 Q6W5P4 2/20 0.35
POLB P06746 2/20 0.35
ALDH1A1 P00352 1/20 0.35
RECQL P46063 1/20 0.35
PAX8 Q06710 1/20 0.35
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7339287 0.77 ITGA4 (0.39) LTA4HITGA4ITGB7MEN1KMT2A
SCHEMBL2059438 0.77 ITGA4 (0.42) LTA4HITGA4ITGB7ATMSLC7A5
SCHEMBL9052981 0.76 ITGA4 (0.45) LTA4HLAP3SLC15A1ITGA4ITGB7
SCHEMBL1519895 0.76 SLC7A5 (0.41) LTA4HLAP3ITGA4ITGB7ATM
SCHEMBL28301558 0.76 ADRA2A (0.40) MEN1KMT2AATML3MBTL1MAPT
SCHEMBL7339280 0.76 KLK5 (0.53) MEN1KMT2APKMATMNPSR1
SCHEMBL11027685 0.75 SLC7A5 (0.46) LTA4HLAP3SLC15A1ITGA4ITGB7
SCHEMBL7369988 0.75 PPARG (0.38) LTA4HITGA4ITGB7MEN1KMT2A
SCHEMBL5650824 0.75 ATM (0.38) LTA4HKMT2AATML3MBTL1SLC7A5
SCHEMBL5652634 0.75 ATM (0.38) LTA4HKMT2AATML3MBTL1SLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed