SCHEMBL7339381

SCHEMBL7339381

COc1cc(-c2ccccc2)ccc1CC(N)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TPH1 P17752 4/20 0.47
SLC1A5 Q15758 1/20 0.46
SLC1A3 P43003 1/20 0.45
SLC1A2 P43004 1/20 0.45
SLC1A1 P43005 1/20 0.45
ALPI P09923 1/20 0.45
PKM P14618 1/20 0.45
PTGS1 P23219 1/20 0.45
XIAP P98170 1/20 0.45
SLC7A5 Q01650 1/20 0.45
GRIA2 P42262 1/20 0.45
NOS3 P29474 1/20 0.45
NOS1 P29475 1/20 0.45
NOS2 P35228 1/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
LMNA P02545 1/20 0.45
MPO P05164 1/20 0.45
MAPT P10636 1/20 0.45
TSHR P16473 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7339373 1.00 TPH1 (0.47) TPH1SLC1A5SLC1A3SLC1A2SLC1A1
Hydrochloric Acid SCHEMBL6505937 0.88 ALDH1A1 (0.46) KDM4EMEN1MAPTKMT2APDCD1
SCHEMBL29750308 0.82 NOS3 (0.55) SLC1A5ALPIPKMPTGS1XIAP
SCHEMBL155234 0.82 NOS3 (0.55) SLC1A5ALPIPKMPTGS1XIAP
SCHEMBL155235 0.82 NOS3 (0.55) SLC1A5ALPIPKMPTGS1XIAP
SCHEMBL4595466 0.82 NOS3 (0.55) SLC1A5ALPIPKMPTGS1XIAP
SCHEMBL5794030 0.81 KDM4E (0.55) TPH1PKMPTGS1SLC7A5GRIA2
SCHEMBL5794029 0.81 KDM4E (0.55) TPH1PKMPTGS1SLC7A5GRIA2
SCHEMBL29519833 0.81 HSD17B10 (0.49) PKMKDM4EMEN1LMNAMAPT
SCHEMBL21803815 0.81 SLC1A5 (0.47) SLC1A5ALPIPKMPTGS1XIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0592367-A2 Phosphono/biaryl substituted dipeptide derivatives CIBA-GEIGY AG (CH) 1994-04-13 EP disclosed
US-5294632-A Diuretics and vasorelaxants CIBA-GEIGY CORPORATION (US) 1994-03-15 US disclosed