SCHEMBL7340274

SCHEMBL7340274

COc1cc(CCC(=O)O)cc2c1OC(NC(=O)CNC(=O)c1cccc(NC=NN)c1)O2

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.39
ITGB3 P05106 2/20 0.35
ITGAV P06756 2/20 0.35
ITGA2B P08514 1/20 0.35
CCR2 P41597 1/20 0.35
ALDH1A1 P00352 4/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
SENP1 Q9P0U3 1/20 0.34
HPGD P15428 2/20 0.34
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34
GPR139 Q6DWJ6 2/20 0.33
TP53 P04637 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6778093 0.89 LMNA (0.43) LMNAITGB3ITGAVITGA2BCCR2
SCHEMBL7340265 0.76 ABCB1 (0.41) LMNAALDH1A1SMN1; SMN2HPGDMAPT
SCHEMBL7343450 0.75 ITGB3 (0.36) LMNAITGB3ITGAVITGA2BALDH1A1
SCHEMBL7346999 0.74 ITGB3 (0.52) ITGB3ITGAVITGA2BALDH1A1SMN1; SMN2
SCHEMBL7338324 0.73 ITGB3 (0.46) LMNAITGB3ITGAVITGA2BALDH1A1
SCHEMBL6777064 0.73 ITGB3 (0.46) LMNAITGB3ITGAVITGA2BALDH1A1
SCHEMBL7349786 0.73 ITGB3 (0.45) LMNAITGB3ITGAVITGA2BALDH1A1
SCHEMBL7837513 0.73 NPC1 (0.38) LMNAALDH1A1SMN1; SMN2MAPTGPR139
SCHEMBL7349108 0.71 ITGB3 (0.38) ITGB3ITGAVITGA2BALDH1A1SENP1
SCHEMBL7348335 0.71 ITGB3 (0.41) LMNAITGB3ITGAVITGA2BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP claimed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO claimed