SCHEMBL7340428

SCHEMBL7340428

CC(C)[C@H](NC(=O)/C=C/Nc1nccs1)C(=O)N[C@@H](Cc1ccccc1)[C@@H](O)[C@H](O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)/C=C/Nc1nccs1)C(C)C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.52
HSPA5 P11021 5/20 0.47
HSPA9 P38646 4/20 0.47
HSPA8 P11142 1/20 0.44
HSPA2 P54652 2/20 0.44
PKM P14618 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
HSPA1A P0DMV8 1/20 0.42
HTT P42858 1/20 0.42
CTSD P07339 3/20 0.41
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
BACE1 P56817 1/20 0.40
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7340432 1.00 CA2 (0.52) CA2HSPA5HSPA9HSPA8HSPA2
SCHEMBL7307572 0.85 CA2 (0.53) CA2HSPA5HSPA9CTSDBACE1
SCHEMBL7307580 0.85 CA2 (0.53) CA2HSPA5HSPA9CTSDBACE1
SCHEMBL6452553 0.79 CA2 (0.62) CA2SMN1; SMN2CTSDTSHRBACE1
SCHEMBL7342544 0.77 CA2 (0.59) CA2SMN1; SMN2CTSDTSHRBACE1
SCHEMBL7342550 0.77 CA2 (0.59) CA2SMN1; SMN2CTSDTSHRBACE1
SCHEMBL7333545 0.76 CA2 (0.54) CA2HSPA5HSPA9PKMCTSD
SCHEMBL7339220 0.76 CA2 (0.71) CA2HSPA5HSPA9CTSDBACE1
SCHEMBL7339662 0.76 CA2 (0.71) CA2HSPA5HSPA9CTSDBACE1
SCHEMBL7339544 0.76 CA2 (0.71) CA2HSPA5HSPA9CTSDBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed