SCHEMBL7340451

SCHEMBL7340451

O=Cc1c[nH]c2cc(F)c(OCc3ccccc3)cc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSV O60911 2/20 0.46
CTSL P07711 2/20 0.46
ERN1 O75460 2/20 0.46
IMPDH2 P12268 2/20 0.43
CYP2A6 P11509 2/20 0.43
MAPT P10636 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CCNB2 O95067 1/20 0.41
CDK1 P06493 1/20 0.41
CDK4 P11802 1/20 0.41
CCNB1 P14635 1/20 0.41
CCND1 P24385 1/20 0.41
CCNB3 Q8WWL7 1/20 0.41
ALDH1A1 P00352 3/20 0.40
HPGD P15428 1/20 0.40
MDH2 P40926 1/20 0.40
KDM4E B2RXH2 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL186998 0.85 IMPDH2 (0.43) IMPDH2CYP2A6MAPTSMN1; SMN2NPC1
SCHEMBL187332 0.85 MAPT (0.44) CTSVCTSLERN1IMPDH2CYP2A6
SCHEMBL187798 0.84 CTSV (0.56) CTSVCTSLERN1IMPDH2CYP2A6
SCHEMBL7823652 0.84 CTSV (0.56) CTSVCTSLERN1IMPDH2CYP2A6
SCHEMBL29957099 0.82 MAPT (0.44) CTSVCTSLERN1IMPDH2CYP2A6
SCHEMBL856019 0.81 ERN1 (0.55) ERN1MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL31113771 0.80 ERN1 (0.54) ERN1MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL1418239 0.78 IMPDH2 (0.61) CTSVCTSLIMPDH2CYP2A6MAPT
SCHEMBL29951517 0.78 IMPDH2 (0.61) CTSVCTSLIMPDH2CYP2A6MAPT
SCHEMBL1791105 0.78 MEN1 (0.60) IMPDH2MAPTSMN1; SMN2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0505322-B1 Aminoguanidines CIBA GEIGY AG (CH) 1998-09-09 EP disclosed
US-5510353-A TREATING IRRITABLE BOWEL SYNDROME, GASTROESOPHAGEAL REFLUX DISEASE, CONSTIPATION, MIGRAINE HEADACHES SANDOZ LTD. (CH) 1996-04-23 US disclosed
EP-0505322-A1 Aminoguanidines SANDOZ LTD. (CH) 1992-09-23 EP disclosed