SCHEMBL7340929

SCHEMBL7340929

CCC(=O)NC1Cc2cccc3c2N(CCC3)C1=O

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 4/20 0.42
MTNR1B P49286 4/20 0.42
CHRM1 P11229 1/20 0.40
CYP1A2 P05177 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALOX15 P16050 1/20 0.40
CES1 P23141 2/20 0.39
HTR1A P08908 3/20 0.39
ACE P12821 3/20 0.39
MME P08473 1/20 0.39
ACE2 Q9BYF1 2/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7341721 0.76 CES1 (0.43) CES1HTR1AACEACE2ALDH1A1
SCHEMBL7353201 0.72 CES1 (0.45) MAPTCES1HTR1AACEMME
SCHEMBL7345026 0.71 AADAT (0.49) CES1HTR1AALDH1A1
SCHEMBL13626167 0.70 ACE (0.49) MTNR1AMTNR1BACEMME
SCHEMBL7353202 0.70 CES1 (0.43) CYP1A2CES1HTR1AALDH1A1CYP3A4
Hydrochloric Acid SCHEMBL7344851 0.70 AADAT (0.48) CES1HTR1AALDH1A1
SCHEMBL7344972 0.70 CES1 (0.38) MTNR1AMTNR1BCES1HTR1AALDH1A1
SCHEMBL13625990 0.68 MTNR1A (0.49) MTNR1AMTNR1BCHRM1CYP1A2MAPT
SCHEMBL4799822 0.68 MTNR1A (0.49) MTNR1AMTNR1BCYP1A2MAPTCYP2C9
SCHEMBL4799807 0.68 MTNR1A (0.49) MTNR1AMTNR1BCYP1A2MAPTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5436240-A Schizophrenia, Parkinson's disease, depression or hypotensive agents using tricyclic amines THE UPJOHN COMPANY (US) 1995-07-25 US disclosed
EP-0480939-B1 HETEROCYCLIC AMINES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY UPJOHN CO (US) 1995-01-25 EP disclosed
US-5273975-A Heterocyclic amines having central nervous system activity THE UPJOHN COMPANY (US) 1993-12-28 US disclosed
WO-1990015058-A1 HETEROCYCLIC AMINES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY THE UPJOHN COMPANY (US) 1990-12-13 WO disclosed