SCHEMBL7353202

SCHEMBL7353202

NC(=O)CCC1Cc2cccc3c2N(CCC3)C1=O

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.43
NPC1 O15118 1/20 0.36
TTR P02766 1/20 0.36
HTR1A P08908 3/20 0.35
ACHE P22303 2/20 0.35
MEN1 O00255 2/20 0.34
GAA P10253 2/20 0.34
KMT2A Q03164 2/20 0.34
ALDH1A1 P00352 2/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
RIPK1 Q13546 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7353201 0.78 CES1 (0.45) CES1HTR1AMEN1KMT2AALDH1A1
SCHEMBL7345026 0.74 AADAT (0.49) CES1HTR1AMEN1GAAKMT2A
Hydrochloric Acid SCHEMBL7344851 0.73 AADAT (0.48) CES1HTR1AMEN1GAAKMT2A
SCHEMBL6338659 0.73 DRD2 (0.43) CES1HTR1AACHE
SCHEMBL7340929 0.70 MTNR1A (0.42) CES1HTR1AALDH1A1CYP1A2CYP3A4
SCHEMBL7341721 0.67 CES1 (0.43) CES1HTR1AMEN1GAAKMT2A
SCHEMBL988203 0.66 CES1 (0.56) CES1NPC1TTRMEN1GAA
SCHEMBL1762224 0.64 CES1 (0.57) CES1
SCHEMBL3133027 0.63 CES1 (0.46) CES1HTR1AMEN1GAAKMT2A
SCHEMBL9560034 0.62 CES1 (0.50) CES1NPC1TTRHTR1AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1990015058-A1 HETEROCYCLIC AMINES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY THE UPJOHN COMPANY (US) 1990-12-13 WO disclosed