SCHEMBL7340943

SCHEMBL7340943

NN=CNc1cccc(C(=O)NCC(=O)NC2(Br)C=C(Cl)C=C(CCC(=O)O)C2)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 4/20 0.34
ITGA5 P08648 4/20 0.34
KMT2A Q03164 2/20 0.34
ITGB3 P05106 4/20 0.33
ITGAV P06756 3/20 0.33
MDM4 O15151 2/20 0.33
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
ITGA2B P08514 1/20 0.31
GPR139 Q6DWJ6 2/20 0.31
MEN1 O00255 1/20 0.31
ATM Q13315 1/20 0.31
KDM4E B2RXH2 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
MDM2 Q00987 2/20 0.31
PPARG P37231 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
GRK2 P25098 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7348232 0.91 ITGB3 (0.33) ITGB1ITGA5KMT2AITGB3ITGAV
SCHEMBL7348831 0.90 ITGB3 (0.33) ITGB1ITGA5KMT2AITGB3ITGAV
SCHEMBL7340934 0.88 ITGB3 (0.37) ITGB1ITGA5KMT2AITGB3ITGAV
SCHEMBL7346234 0.82 KMT2A (0.34) ITGB1ITGA5KMT2AITGB3ITGAV
SCHEMBL7341130 0.82 KMT2A (0.35) ITGB1ITGA5KMT2AITGB3ITGAV
SCHEMBL7347263 0.81 ITGB3 (0.34) ITGB1ITGA5ITGB3ITGAVMDM4
SCHEMBL7341076 0.80 SMN1; SMN2 (0.36) KMT2AITGB3ITGAVALDH1A1ITGA2B
SCHEMBL7403130 0.79 HTT (0.36) ITGB1ITGA5ITGB3ITGAVGPR139
SCHEMBL7348225 0.79 ITGB3 (0.38) ITGB1KMT2AITGB3ITGAVITGA2B
SCHEMBL7348610 0.79 ITGB3 (0.33) ITGB1ITGA5KMT2AITGB3ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP claimed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO claimed