SCHEMBL7342196

SCHEMBL7342196

CC(C)(C)[Si](C)(C)OC1CCC2(CCC(/C=C/c3cccnc3)CC2)CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.35
PTGS2 P35354 3/20 0.35
ALOX5 P09917 2/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
PTAFR P25105 1/20 0.33
NPC1 O15118 4/20 0.32
RAB9A P51151 4/20 0.32
KDM4E B2RXH2 1/20 0.32
JUN P05412 1/20 0.32
MAPT P10636 1/20 0.32
NFKB1 P19838 1/20 0.32
MAPK1 P28482 1/20 0.32
GPR55 Q9Y2T6 1/20 0.32
LMNA P02545 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7343297 1.00 PTGS1 (0.35) PTGS1PTGS2ALOX5CYP11B1CYP11B2
SCHEMBL7342205 1.00 PTGS1 (0.35) PTGS1PTGS2ALOX5CYP11B1CYP11B2
SCHEMBL7340227 0.77 CYP11B1 (0.42) PTGS1PTGS2ALOX5CYP11B1CYP11B2
SCHEMBL7340223 0.77 CYP11B1 (0.42) PTGS1PTGS2ALOX5CYP11B1CYP11B2
SCHEMBL7345200 0.77 CYP11B1 (0.42) PTGS1PTGS2ALOX5CYP11B1CYP11B2
SCHEMBL27802133 0.73 CYP11B1 (0.57) PTGS1PTGS2ALOX5CYP11B1CYP11B2
SCHEMBL7340708 0.72 CHRNB2 (0.43) PTGS2NPC1CHRNB2CHRNA4
SCHEMBL7340701 0.72 CHRNB2 (0.43) PTGS2NPC1CHRNB2CHRNA4
SCHEMBL7348148 0.72 CHRNB2 (0.43) PTGS2NPC1CHRNB2CHRNA4
SCHEMBL5949116 0.72 NFE2L2 (0.40) PTGS1PTGS2ALOX5NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0578080-B1 3,9-disubstituted-spiro (5.5)undecanes active on the cardiovascular system, process for their preparation and pharmaceutical composition containing same SIGMA TAU IND FARMACEUTI (IT) 1997-04-23 EP disclosed
US-5444082-A Treats hypertension and heart failure SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A. (IT) 1995-08-22 US disclosed
EP-0578080-A2 3,9-disubstituted-spiro (5.5)undecanes active on the cardiovascular system, process for their preparation and pharmaceutical composition containing same Sigma-Tau Industrie Farmaceutiche Riunite S.p.A. (IT) 1994-01-12 EP disclosed