SCHEMBL734246

SCHEMBL734246

OCCn1ccc2ccccc21

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 4/20 0.76
CCND1 P24385 4/20 0.76
LMNA P02545 1/20 0.61
HTR2A P28223 1/20 0.59
HTR2C P28335 1/20 0.59
KMT2A Q03164 2/20 0.56
MAPK1 P28482 2/20 0.56
HTT P42858 1/20 0.51
ALDH1A1 P00352 2/20 0.51
TSHR P16473 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
MEN1 O00255 1/20 0.51
MAPT P10636 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C19 P33261 1/20 0.51
MTNR1A P48039 1/20 0.50
MTNR1B P49286 1/20 0.50
HSD17B10 Q99714 1/20 0.50
HTR6 P50406 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30063707 1.00 CDK4 (0.76) CDK4CCND1LMNAHTR2AHTR2C
Alcohol SCHEMBL734139 0.94 CDK4 (0.68) CDK4CCND1LMNAHTR2AHTR2C
SCHEMBL30701168 0.88 CDK4 (0.78) CDK4CCND1LMNAHTR2AHTR2C
SCHEMBL4992403 0.88 CDK4 (0.78) CDK4CCND1LMNAHTR2AHTR2C
SCHEMBL11366447 0.87 CDK4 (1.00) CDK4CCND1LMNAHTR2AHTR2C
SCHEMBL24398975 0.85 CDK4 (0.82) CDK4CCND1LMNAHTR2AHTR2C
SCHEMBL1293253 0.85 CDK4 (0.82) CDK4CCND1LMNAHTR2AHTR2C
SCHEMBL29368287 0.85 CDK4 (0.82) CDK4CCND1LMNAHTR2AHTR2C
SCHEMBL2076869 0.83 CDK4 (0.68) CDK4CCND1LMNAHTR2AHTR2C
SCHEMBL30342074 0.83 CDK4 (0.68) CDK4CCND1LMNAHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 145 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110776497-B Preparation method for constructing two-dimensional organic layer based on cation-pi interaction 西北工业大学 2022-12-13 CN claimed
CN-110776497-A Preparation method for constructing two-dimensional organic layer based on cation-pi interaction 西北工业大学 2020-02-11 CN claimed
CN-101824027-B Polysubstituted tetrahydroquinoline derivative with optical activity and synthetic method and use thereof UNIV BEIJING 2013-09-04 CN claimed
EP-2317849-A1 METHOD FOR TREATING PULMONARY DISEASES USING RHO KINASE INHIBITOR COMPOUNDS Inspire Pharmaceuticals, Inc. (US) 2011-05-11 EP claimed
CN-101824027-A Polysubstituted tetrahydroquinoline derivative with optical activity and synthetic method and use thereof UNIV BEIJING 2010-09-08 CN claimed
JP-2110107-A None JP disclosed
CN-117024759-A Organic Pt metal macrocyclic group two-dimensional supermolecule assembly constructed based on oriented cation-pi action, and preparation method and application thereof 陕西中医药大学 2023-11-10 CN disclosed
WO-2023141595-A2 FUNCTIONALIZED ALKYLAMINES TERRAN BIOSCIENCES, INC. (US) 2023-07-27 WO disclosed
EP-3298003-B1 BENZOIMIDAZOLE DERIVATIVES AS PAD4 INHIBITORS GLAXOSMITHKLINE IP DEV LTD (GB) 2023-04-19 EP disclosed
EP-3298003-B1 BENZOIMIDAZOLE DERIVATIVES AS PAD4 INHIBITORS GLAXOSMITHKLINE IP DEV LTD (GB) 2023-04-19 EP disclosed
CN-110776497-B Preparation method for constructing two-dimensional organic layer based on cation-pi interaction 西北工业大学 2022-12-13 CN disclosed
EP-3472162-B1 HETEROARYL ESTROGEN RECEPTOR MODULATORS AND USES THEREOF HOFFMANN LA ROCHE (CH) 2021-11-17 EP disclosed
EP-0061333-B1 9-(2-(3-INDOLYL)ETHYL)-1-OXA-4,9-DIAZASPIRO(5.5)UNDECAN-3-ONES SYNTEX (U.S.A.) INC. (US) 1986-01-02 EP disclosed
EP-0022634-B1 ACYLATED INDOLE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS AND DRUGS COMPRISING THEM TEIJIN LIMITED (JP) 1983-04-06 EP disclosed
EP-0061333-A1 9-(2-(3-Indolyl)ethyl)-1-oxa-4,9-diazaspiro(5.5)undecan-3-ones SYNTEX (U.S.A.) INC. (US) 1982-09-29 EP disclosed
US-4332804-A TREATMENT OF HYPERTENSION, CONGESTIVE HEART FAILURE, ARRHYTHMIA, MIGRAINE, VASOSPASTIC DISORDERS AND ASTHMA SYNTEX (U.S.A.) INC. (US) 1982-06-01 US disclosed
EP-0022634-A1 Acylated indole derivatives, processes for their preparation and pharmaceutical compositions and drugs comprising them TEIJIN LIMITED (JP) 1981-01-21 EP disclosed
US-4066763-A Thiazinoindoles useful as antidepressants AYERST MCKENNA AND HARRISON LTD. (CA) 1978-01-03 US disclosed
US-4012511-A ANTIULCER AGENTS AYERST MCKENNA & HARRISON LTD. (CA) 1977-03-15 US disclosed
US-3962236-A ANTIDEPRESSANTS, ANTI-ULCER AYERST MCKENNA AND HARRISON LTD. (CA) 1976-06-08 US disclosed