SCHEMBL7344227

SCHEMBL7344227

NN=CNc1cccc(C(=O)NCC(=O)NOC(=O)CCC(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GPR139 Q6DWJ6 3/20 0.37
CCR2 P41597 2/20 0.36
MAPK1 P28482 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
TAAR1 Q96RJ0 1/20 0.36
EPHX2 P34913 1/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 3/20 0.34
MEN1 O00255 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7344218 0.84 HTT (0.46) HTTL3MBTL1CCR2EPHX2GAA
SCHEMBL7344242 0.79 GPR139 (0.44) HTTL3MBTL1GPR139SMN1; SMN2TAAR1
SCHEMBL7339304 0.77 ITGB3 (0.45) HTTL3MBTL1GPR139KMT2AMEN1
SCHEMBL27502755 0.75 ITGB3 (0.41) HTTL3MBTL1SMN1; SMN2TAAR1EPHX2
SCHEMBL7344443 0.75 GPR139 (0.41) HTTL3MBTL1GPR139CCR2SMN1; SMN2
SCHEMBL7347755 0.74 ITGB3 (0.43) GPR139GAA
SCHEMBL6780118 0.74 ITGB3 (0.47) HTTL3MBTL1GPR139KMT2AMEN1
SCHEMBL7346999 0.73 ITGB3 (0.52) HTTL3MBTL1SMN1; SMN2GAAALDH1A1
SCHEMBL6779680 0.73 GPR139 (0.45) GPR139MAPK1KMT2AMEN1
SCHEMBL7347064 0.72 GPR139 (0.46) HTTL3MBTL1GPR139CCR2EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP claimed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO claimed