SCHEMBL7344244

SCHEMBL7344244

NC1CNc2c(cc(Br)cc2[N+](=O)[O-])C1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.38
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
ERN1 O75460 1/20 0.34
S100A4 P26447 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
CYP3A4 P08684 1/20 0.31
GALR3 O60755 1/20 0.31
THRB P10828 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
GPR35 Q9HC97 1/20 0.30
TYMS P04818 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7343407 0.99 AKR1B1 (0.37) AKR1B1ALDH1A1MAPTERN1S100A4
SCHEMBL7346523 0.80 AKR1B1 (0.36) AKR1B1ALDH1A1MAPTERN1S100A4
SCHEMBL7344187 0.77 AKR1B1 (0.34) AKR1B1ALDH1A1MAPTERN1HTR2A
SCHEMBL7349533 0.76 AKR1B1 (0.37) AKR1B1ALDH1A1MAPTERN1S100A4
SCHEMBL13090518 0.76 AKR1B1 (0.37) AKR1B1ALDH1A1MAPTERN1S100A4
SCHEMBL27819557 0.75 AKR1B1 (0.36) AKR1B1ALDH1A1MAPTERN1S100A4
Hydrochloric Acid SCHEMBL2839862 0.75 AKR1B1 (0.36) AKR1B1ALDH1A1MAPTERN1S100A4
SCHEMBL7341794 0.75 FYN (0.38) ALDH1A1CYP3A4
SCHEMBL7351948 0.75 DRD2 (0.33) AKR1B1ALDH1A1MAPT
SCHEMBL768764 0.74 ALDH1A1 (0.54) AKR1B1ALDH1A1MAPTERN1S100A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5436240-A Schizophrenia, Parkinson's disease, depression or hypotensive agents using tricyclic amines THE UPJOHN COMPANY (US) 1995-07-25 US disclosed
EP-0480939-B1 HETEROCYCLIC AMINES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY UPJOHN CO (US) 1995-01-25 EP disclosed
US-5273975-A Heterocyclic amines having central nervous system activity THE UPJOHN COMPANY (US) 1993-12-28 US disclosed
EP-0480939-A1 HETEROCYCLIC AMINES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY. UPJOHN CO (US) 1992-04-22 EP disclosed
WO-1990015058-A1 HETEROCYCLIC AMINES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY THE UPJOHN COMPANY (US) 1990-12-13 WO disclosed